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科研机构
大连化学物理研究所 [2]
浙江工商大学 [2]
上海药物研究所 [1]
上海大学 [1]
湖南农业大学 [1]
复旦大学上海医学院 [1]
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期刊论文 [10]
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miR-21 enhances the protective effect of loperamide on rat cardiomyocytes against hypoxia/reoxygenation, reactive oxygen species production and apoptosis via regulating Akap8 and Bard1 expression
期刊论文
EXPERIMENTAL AND THERAPEUTIC MEDICINE, 2019, 卷号: 17, 期号: 2
作者:
Shen, Hong
;
Yao, Zhifeng
;
Zhao, Weipeng
;
Zhang, Yaping
;
Yao, Chenling
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/12/05
loperamide
miR-21
hypoxia
reoxygenation
cardiomyocytes
Comparative metabolism of DDAO benzoate in liver microsomes from various species
期刊论文
TOXICOLOGY IN VITRO, 2017, 卷号: 44, 页码: 280-286
作者:
Ge, Guang-Bo
;
Ma, Hong-Ying
;
Yang, Jia-Da
;
Hou, Jie
;
Zou, Li-Wei
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2017/12/19
DDAB hydrolysis
Carboxylesterase 2 (CE2)
Species differences
Liver microsomes
Comparative metabolism of DDAO benzoate in liver microsomes from various species
期刊论文
TOXICOLOGY IN VITRO, 2017, 卷号: 44, 页码: 280-286
作者:
Ma, Hong-Ying
;
Yang, Jia-Da
;
Hou, Jie
;
Zou, Li-Wei
;
Jin, Qiang
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2017/12/19
DDAB hydrolysis
Carboxylesterase 2 (CE2)
Species differences
Liver microsomes
Loperamide inhibits sodium channels to alleviate inflammatory hyperalgesia
期刊论文
2017, 卷号: 117, 页码: 282-291
作者:
Wu Ying
;
Zou Beiyan
;
Liang Lingli
;
Li Min
;
Tao Yuan-Xiang
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2020/01/04
Loperamide
Opioid receptor
Pain
Nav1.7
Sodium channel
Identification of novel small-molecule inhibitors targeting menin-MLL interaction, repurposing the antidiarrheal loperamide
期刊论文
ORGANIC & BIOMOLECULAR CHEMISTRY, 2016, 卷号: 14, 期号: 36, 页码: 8503-8519
作者:
Yue, Liyan
;
Du, Juanjuan
;
Ye, Fei
;
Chen, Zhifeng
;
Li, Lianchun
收藏
  |  
浏览/下载:26/0
  |  
提交时间:2019/01/08
Magnolol and honokiol regulate the calcium-activated potassium channels signaling pathway in Enterotoxigenic Escherichia coli-induced diarrhea mice
期刊论文
European Journal of Pharmacology, 2015, 卷号: 755, 页码: 66-73
作者:
Deng, Yanli
;
Han, Xuefeng
;
Tang, Shaoxun
;
Xiao, Wenjun*
;
Tan, Zhiliang
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2019/12/23
CaM
calmodulin 1
CaMKIIα
calcium/calmodulin-dependent protein kinase II alpha subunit
CaMKIIβ
calcium/calmodulin-dependent protein kinase II beta subunit
PKC
protein kinase C
IP3
inositol 1,4,5-trisphosphate
SK
potassium intermediate/small conductance calcium-activated channels
BKα1
potassium large conductance calcium-activated channel, subfamily M, alpha member 1
BKβ
potassium large conductance calcium-activated channel, subfamily M, beta.
Magnolol (PubChem CID: 72300)
Honokiol ( PubChem CID: 72303)
Loperamide hydrochloride ( PubChem CID: 71420)
Magnolol
Honokiol
Diarrhea
Enterotoxigenic Escherichia coli
Calcium-activated potassium channel
Inositol 1,4,5-trisphosphate receptor
Discovery of loperamide as an antagonist of angiopoietin1 and angiopoietin2 by virtual screening
期刊论文
2012, 卷号: 22, 期号: 7, 页码: 2388
作者:
Gong, Xing Wen[1]
;
Mai, Jun Hua[2]
;
Xu, Yu Hong[2]
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2019/12/26
Loperamide, an antidiarrhea drug, has antitumor activity by inducing cell apoptosis
期刊论文
2012, 卷号: 65, 期号: 3, 页码: 372
作者:
Gong, Xing Wen[1]
;
Xu, Yu Hong[2]
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2019/12/26
Traditional Chinese formula, lubricating gut pill, improves loperamide-induced rat constipation involved in enhance of Cl- secretion across distal colonic epithelium
期刊论文
JOURNAL OF ETHNOPHARMACOLOGY, 2010, 卷号: 130, 期号: 2
作者:
Wu, Dazheng
;
Wang, Xinhong
;
Zhou, Jiyan
;
Yuan, Jianye
;
Cui, Bo
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2019/12/05
Colonic epithelium
Lubricating gut pill
Cl- secretion
Constipation
Laxative effect
Traditional Chinese formula, lubricating gut pill, improves loperamide-induced rat constipation involved in enhance of Cl- secretion across distal colonic epithelium
期刊论文
Journal of ethnopharmacology, 2010, 卷号: 130, 页码: 347-53
作者:
Wu Dazheng[1]
;
Wang Xinhong[2]
;
Zhou Jiyan[3]
;
Yuan Jianye[4]
;
Cui Bo[5]
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2019/04/30
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