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SAF-248, a novel PI3K delta-selective inhibitor, potently suppresses the growth of diffuse large B-cell lymphoma 期刊论文
ACTA PHARMACOLOGICA SINICA, 2021, 页码: 11
作者:  Zhang, Xi;  Duan, Yu-ting;  Wang, Yi;  Zhao, Xing-dong;  Sun, Yi-ming
收藏  |  浏览/下载:37/0  |  提交时间:2021/05/24
B591, a novel specific pan-PI3K inhibitor, preferentially targets cancer stem cells 期刊论文
ONCOGENE, 2019, 卷号: 38, 期号: 18, 页码: 3371-3386
作者:  Zhou, Hongyu;  Yu, Chunlei;  Kong, Lingmei;  Xu, Xiaoliang;  Yan, Juming
收藏  |  浏览/下载:191/0  |  提交时间:2019/06/24
Identification, structure modification, and characterization of potential small-molecule SGK3 inhibitors with novel scaffolds 期刊论文
Acta pharmacologica Sinica, 2018, 卷号: 39, 期号: 12, 页码: 1902-1912
作者:  Gong, Grace Qun;  Wang, Ke;  Dai, Xin-Chuan;  Zhou, Yan;  Basnet, Rajesh
收藏  |  浏览/下载:98/0  |  提交时间:2019/01/08
Synthesis, biological evaluation and structure-activity relationship of a novel class of PI3K alpha H1047R mutant inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 158, 页码: 707-719
作者:  Zhang, Ning;  Yu, Zhimei;  Yang, Xiaohong;  Zhou, Yan;  Wang, Jia
收藏  |  浏览/下载:85/0  |  提交时间:2019/01/08
Discovery of (S)-2-amino-N-(5-(6-chloro-5-(3-methylphenylsulfonamido)pyridin-3-yl)-4-methylthiazol-2-yl)-3-methylbutanamide (CHMFL-PI3KD-317) as a potent and selective phosphoinositide 3-kinase delta (PI3K delta) inhibitor 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 156, 页码: 831-846
作者:  Liang, Xiaofei;  Li, Feng;  Chen, Cheng;  Jiang, Zongru;  Wang, Aoli
收藏  |  浏览/下载:13/0  |  提交时间:2019/12/10
identificationstructuremodificationandcharacterizationofpotentialsmallmoleculesgk3inhibitorswithnovelscaffolds 期刊论文
中国药理学报英文版, 2018, 卷号: 039, 期号: 012, 页码: 1902
作者:  Grace Qun Gong;  Ke Wang;  XinChuan Dai;  Yan Zhou;  Rajesh Basnet
收藏  |  浏览/下载:4/0  |  提交时间:2020/07/01
Pharmacologic characterization of SHR8443, a novel dual inhibitor of phosphatidylinositol 3-kinase and mammalian target of rapamycin 期刊论文
ONCOTARGET, 2017, 卷号: 8, 期号: 64, 页码: 107977-107990
作者:  Xie, Chengying;  Chen, Xiangling;  Zheng, Mingyue;  Liu, Xiaohong;  Wang, Hongbin
收藏  |  浏览/下载:27/0  |  提交时间:2019/01/08
G beta 1 is required for neutrophil migration in zebrafish 期刊论文
DEVELOPMENTAL BIOLOGY, 2017, 卷号: 428, 期号: 1, 页码: 135-147
作者:  Ke, Wenfan;  Ye, Ding;  Mersch, Kacey;  Xu, Hui;  Chen, Songhai
收藏  |  浏览/下载:16/0  |  提交时间:2019/09/17
Puquitinib, a novel orally available PI3K inhibitor, exhibits potent antitumor efficacy against acute myeloid leukemia 期刊论文
CANCER SCIENCE, 2017, 卷号: 108, 期号: 7, 页码: 1476-1484
作者:  Xie, Chengying;  He, Ye;  Zhen, Mingyue;  Wang, Yulan;  Xu, Yongping
收藏  |  浏览/下载:18/0  |  提交时间:2019/01/08
Molecular Mechanism Of Carcinoembryonic Antigen-Related Cell Adhesion Molecule 1 Isoforms-Regulated Inflammation Response In Acute Exacerbation Of Chronic Obstructive Pulmonary Disease 会议论文
作者:  Zhu, Y.;  Wang, X.
收藏  |  浏览/下载:3/0  |  提交时间:2019/12/05


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