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科研机构
上海药物研究所 [4]
厦门大学 [2]
北京大学 [2]
清华大学 [1]
金属研究所 [1]
昆明植物研究所 [1]
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期刊论文 [14]
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2019 [3]
2016 [3]
2014 [1]
2012 [2]
2010 [1]
2009 [2]
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Ultra-long silver nanowires induced mitotic abnormalities and cytokinetic failure in A549 cells
期刊论文
NANOTOXICOLOGY, 2019, 卷号: 13, 期号: 4, 页码: 543-557
作者:
Wang, Fengbang
;
Chen, Ying
;
Wang, Yuanyuan
;
Yin, Yongguang
;
Qu, Guangbo
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2020/10/22
Ultra-long silver nanowires
mitotic abnormalities
cytokinetic failure
multinucleation
ROS
Antiproliferative Aspidosperma-Type Monoterpenoid Indole Alkaloids from Bousigonia mekongensis Inhibit Tubulin Polymerization
期刊论文
MOLECULES, 2019, 卷号: 24, 期号: 7, 页码: 10
作者:
Zhang, Yu
;
Goto, Masuo
;
Oda, Akifumi
;
Hsu, Pei-Ling
;
Guo, Ling-Li
收藏
  |  
浏览/下载:67/0
  |  
提交时间:2019/07/29
aspidosperma-type
monoterpenoid indole alkaloids
antiproliferative activity
tubulin inhibitor
Bousigonia mekongensis
Synthetic derivatives of the natural product 13-amino 2-desoxy-4-epi-pulchellin inhibit STAT3 signaling and induce G2/M arrest and death of colon cancer cells
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 卷号: 29, 期号: 6, 页码: 782-785
作者:
Niu, Junxing
;
Huang, Hui
;
Wang, Fei
;
Zhang, Xianjing
;
Liu, Yi
收藏
  |  
浏览/下载:31/0
  |  
提交时间:2020/07/01
Sesquiterpene-lactone
JAK2/STAT3
Michael addition reaction
Antitumor
Colorectal carcinoma
Moderate intensity static magnetic fields affect mitotic spindles and increase the antitumor efficacy of 5-FU and Taxol
期刊论文
BIOELECTROCHEMISTRY, 2016, 卷号: 109, 期号: 无, 页码: 31-40
作者:
Luo, Yan
;
Ji, Xinmiao
;
Liu, Juanjuan
;
Li, Zhiyuan
;
Wang, Wenchao
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2017/11/10
Static Magnetic Field
Microtubule
Mitosis
Cancer Cells
5-fluorouracil
Cisplatin
Identification of acylthiourea derivatives as potent Plk1 PBD inhibitors
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016
Yun, Taikangxiang
;
Qin, Tan
;
Liu, Ying
;
Lai, Luhua
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2017/12/04
Polo-like kinase 1
Polo-box domain
Small molecular inhibitor
Halogenosulfamoylphenyl acylthiourea
Binding affinity
In vitro assay
POLO-LIKE KINASE
INDUCE MITOTIC ARREST
BOX DOMAIN
PROGNOSTIC-SIGNIFICANCE
CANCER-CELLS
TUMOR-CELLS
DRUG DESIGN
EXPRESSION
DISCOVERY
DOCKING
Discovery of Novel Polo-Like Kinase 1 Polo-Box Domain Inhibitors to Induce Mitotic Arrest in Tumor Cells
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2016
Qin, Tan
;
Chen, Fangjin
;
Zhuo, Xiaolong
;
Guo, Xiao
;
Yun, Taikangxiang
;
Liu, Ying
;
Zhang, Chuanmao
;
Lai, Luhua
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2017/12/04
ADVANCED SOLID MALIGNANCIES
GROWTH IN-VIVO
PHASE-I
CELLULAR UPTAKE
PLK1
POLO-LIKE-KINASE-1
CANCER
PHOSPHOPEPTIDES
IDENTIFICATION
RECOGNITION
Mitotic DNA damages induced by carbon-ion radiation incur additional chromosomal breaks in polyploidy
期刊论文
TOXICOLOGY LETTERS, 2014, 卷号: 230, 页码: 36-47
作者:
Liu, XG
;
Ye, F
;
Zhao, T
;
Jin, XD
;
Liu, XX
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2015/11/20
Induced Cell-death
Histone H2ax
Cancer-cells
Mammalian-cells
Tumor-cells
Apoptosis
Catastrophe
P53
Phosphorylation
Irradiation
A Cell-Based Assay for Screening Spindle Checkpoint Inhibitors
期刊论文
2012
Wu, Zhen Hua
;
Hu, Long Yu
;
Xu, Da Qian
;
许大千
;
Li, Xiaotong
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2013/03/01
MITOTIC CHECKPOINT
ASSEMBLY CHECKPOINT
AURORA KINASES
CANCER-CELLS
FREQUENT IMPAIRMENT
HIGH-THROUGHPUT
MAD2
ANAPHASE
GENES
INSTABILITY
Discovery of Novel 2-N-Aryl-Substituted Benzenesulfonamidoacetamides: Orally Bioavailable Tubulin Polymerization Inhibitors with Marked Antitumor Activities
期刊论文
CHEMMEDCHEM, 2012, 卷号: 7, 期号: 4, 页码: 680-693
作者:
Liu, Zulong
;
Zhou, Zuyu
;
Tian, Wei
;
Fan, Xing
;
Xue, Ding
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2019/01/08
antitumor agents
benzenesulfonamidoacetamides
bioactive compounds
screening
tubulin
NuSAP is degraded by APC/C-Cdh1 and its overexpression results in mitotic arrest dependent of its microtubules' affinity
期刊论文
2010, 2010, OCT
Li, Lu
;
Zhou, Ying
;
Sun, Libo
;
Xing, Guichun
;
Tian, Chunyan
;
Sun, Jing
;
Zhang, Lingqiang
;
He, Fuchu
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2017/06/15
NuSAP
APC/C
mitotic arrest
degradation
ANAPHASE-PROMOTING COMPLEX
CELL-CYCLE CONTROL
SPINDLE CHECKPOINT
AURORA-B
KEN-BOX
DEGRADATION
ANEUPLOIDY
PROTEIN
EXIT
COMPLEX/CYCLOSOME
Cell Biology
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