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上海药物研究所 [7]
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厦门大学 [2]
北京大学 [2]
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期刊论文 [22]
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Endosulfan promotes cell migration via PTP4A3-mediated signaling pathways in HUVECs
期刊论文
ECOTOXICOLOGY AND ENVIRONMENTAL SAFETY, 2020, 卷号: 192, 页码: 1-9
作者:
Li, Heng
;
Liu, Shiqi
;
Hu, Yumeng
;
Zhao, Bin
;
Sun, Yeqing
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2021/09/14
Endosulfan
Cell migration
PTP4A3
Signaling pathway
Endothelial cells
Novel selective TOPK inhibitor SKLB-C05 inhibits colorectal carcinoma growth and metastasis
期刊论文
Cancer Letters, 2019, 卷号: Vol.445, 页码: 11-23
作者:
Tiantao Gao
;
Quanfang Hu
;
Xi Hu
;
Qian Lei
;
Zhanzhan Feng
收藏
  |  
浏览/下载:68/0
  |  
提交时间:2019/02/25
MAPK
signaling
pathway
Mitosis
failure
DNA-reparation
failure
FAK
signaling
Apoptosis
Structure-based modification of carbonyl-diphenylpyrimidines (Car-DPPYs) as a novel focal adhesion kinase (FAK) inhibitor against various stubborn cancer cells
期刊论文
2019, 卷号: 172, 页码: 154-162
作者:
Wang, Luhong
;
Ai, Min
;
Yu, Jiawen
;
Jin, Lingling
;
Wang, Changyuan
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2020/01/03
Cancer
FAK
Inhibitor
Pyrimidine
Activity
CTC clusters induced by heparanase enhance breast cancer metastasis
期刊论文
ACTA PHARMACOLOGICA SINICA, 2018, 卷号: 39, 期号: 8, 页码: 1326-1337
作者:
Wei, Rong-rui
;
Sun, Dan-ni
;
Yang, Hong
;
Yan, Juan
;
Zhang, Xiong
收藏
  |  
浏览/下载:89/0
  |  
提交时间:2019/01/08
human breast cancer
CTC clusters
heparanase
metastasis
cell adhesion
adhesion molecules
suspension culture method
New microtubulin inhibitor MT189 suppresses angiogenesis via the JNK-VEGF/VEGFR2 signaling axis
期刊论文
CANCER LETTERS, 2018, 卷号: 416, 页码: 57-65
作者:
Xu, Lin
;
Wang, Wei
;
Meng, Tao
;
Ma, Lan-Ping
;
Tong, Lin-Jiang
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2019/01/08
MT189
Microtubulin inhibitor
VEGF
Src
JNK
Cell adhesion
Space microgravity drives transdifferentiation of human bone marrow-derived mesenchymal stem cells from osteogenesis to adipogenesis
期刊论文
FASEB JOURNAL, 2018, 卷号: 32, 期号: 8, 页码: 4444-4458
作者:
Zhang, Cui
;
Li, Liang
;
Jiang, Yuanda
;
Wang, Cuicui
;
Geng, Baoming
收藏
  |  
浏览/下载:49/0
  |  
提交时间:2018/09/06
Hmscs
Signaling Pathway
Sj-10 Satellite
Rna-seq
Structure Optimization and Structure-Activity Relationship Study of a Kind of Type II FAK Inhibitors with N-Phenylpyrazole Ureas
期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2018, 卷号: 38, 期号: 11
作者:
Gong Chaochao
;
Tan Hanyi
;
Zhang Qian
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2019/12/05
focal adhesion kinase
allosteric hydrophobic pocket
type II inhibitor
N-phenylpyrazole
structure optimization
RN1, a novel galectin-3 inhibitor, inhibits pancreatic cancer cell growth in vitro and in vivo via blocking galectin-3 associated signaling pathways
期刊论文
ONCOGENE, 2017, 卷号: 36, 期号: 9, 页码: 1297-1308
作者:
Zhang, L.
;
Wang, P.
;
Qin, Y.
;
Cong, Q.
;
Shao, C.
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2019/01/08
PTK2-mediated degradation of ATG3 impedes cancer cells susceptible to DNA damage treatment
期刊论文
AUTOPHAGY, 2017
Ma, Ke
;
Fu, Wan
;
Tang, Ming
;
Zhang, Chaohua
;
Hou, Tianyun
;
Li, Ran
;
Lu, Xiaopeng
;
Wang, Yanan
;
Zhou, Jingyi
;
Li, Xue
;
Zhang, Luyao
;
Wang, Lina
;
Zhao, Ying
;
Zhu, Wei-Guo
收藏
  |  
浏览/下载:10/0
  |  
提交时间:2017/12/03
ATG3
cancer therapy
mitotic catastrophe
PTK2
tyrosine phosphorylation
FOCAL ADHESION KINASE
MITOTIC CATASTROPHE
AUTOPHAGOSOME FORMATION
OVARIAN-CANCER
TUMOR-GROWTH
FAK
CONJUGATION
CARCINOMA
PATHWAYS
DEATH
Substrate stiffness promotes latent TGF-beta 1 activation in hepatocellular carcinoma
期刊论文
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2017
Pang, Mingshu
;
Teng, Yao
;
Huang, Jianyong
;
Yuan, Yuan
;
Lin, Feng
;
Xiong, Chunyang
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2017/12/03
Hepatocellular carcinoma
Substrate stiffness
Traction forces
Transforming growth factor beta 1
beta 1 integrin
TRANSFORMING GROWTH-FACTOR-BETA-1
EXTRACELLULAR-MATRIX
FOCAL ADHESIONS
BETA
CONTRACTION
FIBROSIS
DISEASE
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