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Rational Design and Evaluation of 6-(Pyrimidin-2-ylamino)-3,4-dihydroquinoxalin-2(1H)-ones as Polypharmacological Inhibitors of BET and Kinases 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 17, 页码: 9787-9802
作者:  Lv, Kaikai;  Chen, Weicong;  Chen, Danqi;  Mou, Jie;  Zhang, Huijie
收藏  |  浏览/下载:12/0  |  提交时间:2020/12/21
Structure-Based Discovery and Development of a Series of Potent and Selective Bromodomain and Extra-Terminal Protein Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 18, 页码: 8642-8663
作者:  Hu, Jianping;  Tian, Chang-Qing;  Damaneh, Mohammadali Soleimani;  Li, Yanlian;  Cao, Danyan
收藏  |  浏览/下载:11/0  |  提交时间:2020/07/01
Structure-based optimization of a series of selective BET inhibitors containing aniline or indoline groups 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 页码: 156-175
作者:  Hu, Jianping;  Wang, Yingqing;  Li, Yanlian;  Cao, Danyan;  Xu, Lin
收藏  |  浏览/下载:34/0  |  提交时间:2019/01/08
Discovery of a series of dihydroquinoxalin-2(1H)-ones as selective BET inhibitors from a dual PLK1-BRD4 inhibitor 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 137, 页码: 176-195
作者:  Hu, Jianping;  Wang, Yingqing;  Li, Yanlian;  Xu, Lin;  Cao, Danyan
收藏  |  浏览/下载:32/0  |  提交时间:2019/01/08
Design, synthesis and evaluation of a novel BRD4 protein inhibitors 期刊论文
Acta Pharmaceutica Sinica, 2017, 卷号: 52, 期号: 10, 页码: 1568-1577
作者:  Hu Jianping;  Li Yanlian;  Shi Huanyu;  Xiong Bing;  Shen Jingkang
收藏  |  浏览/下载:25/0  |  提交时间:2019/01/08
Metal-free tandem cyclization/hydrosilylation to construct tetrahydroquinoxalines 期刊论文
GREEN CHEMISTRY, JAN , 卷号: 20, 期号: 2, 页码: 403-411
作者:  Pan, Yixiao;  Chen, Changjun;  Xu, Xin;  Zhao, Haoqiang;  Han, Jiahong
收藏  |  浏览/下载:8/0  |  提交时间:2018/04/10


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