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科研机构
北京大学 [8]
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期刊论文 [8]
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2017 [1]
2015 [1]
2014 [1]
2012 [3]
2011 [1]
2009 [1]
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专题:北京大学
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Serum polyunsaturated fatty acid metabolites as useful tool for screening potential biomarker of colorectal cancer
期刊论文
PROSTAGLANDINS LEUKOTRIENES AND ESSENTIAL FATTY ACIDS, 2017
Zhang, Li-Jian
;
Chen, Bin
;
Zhang, Jun-jie
;
Li, Jian
;
Yang, Qingjing
;
Zhong, Qi-sheng
;
Zhan, Song
;
Liu, Huwei
;
Cai, Chun
收藏
  |  
浏览/下载:8/0
  |  
提交时间:2017/12/03
Lipidomic
Colorectal cancer
Ultra-high performance liquid chromatography
Mass spectrometry
DRUG-INDUCED APOPTOSIS
CELL LUNG-CANCER
OXIDATIVE STRESS
PPAR-GAMMA
13-HYDROXYOCTADECADIENOIC ACID
PROSTAGLANDIN E-2
ARACHIDONIC-ACID
COLON
GROWTH
15-LIPOXYGENASE-1
Diverse Ways of Perturbing the Human Arachidonic Acid Metabolic Network To Control Inflammation
期刊论文
ACCOUNTS OF CHEMICAL RESEARCH, 2015
Meng, Hu
;
Liu, Ying
;
Lai, Luhua
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2017/12/03
PROSTAGLANDIN E-2 SYNTHASE-1
TRADITIONAL CHINESE MEDICINE
LEUKOTRIENE A(4) HYDROLASE
DUAL INHIBITORS
DRUG DESIGN
LTA(4) HYDROLASE
5-LIPOXYGENASE
DISCOVERY
DERIVATIVES
CYCLOOXYGENASE-2
Benzo[d] isothiazole 1,1-dioxide derivatives as dual functional inhibitors of 5-lipoxygenase and microsomal prostaglandin E-2 synthase-1
期刊论文
生物有机化学与医药化学通讯, 2014
Shang, Erchang
;
Wu, Yiran
;
Liu, Pei
;
Liu, Ying
;
Zhu, Wei
;
Deng, Xiaobing
;
He, Chong
;
He, Shan
;
Li, Cong
;
Lai, Luhua
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2015/11/10
Benzo[d] isothiazole 1,1-dioxide
5-Lipoxygenase
Microsomal prostaglandin E-2 synthase
Dual functional inhibitor
ANTIINFLAMMATORY DRUGS
MPGES-1
BIOLOGY
TARGET
5-LOX
Dynamic Modeling of Human 5-Lipoxygenase-Inhibitor Interactions Helps To Discover Novel Inhibitors
期刊论文
journal of medicinal chemistry, 2012
Wu, Yiran
;
He, Chong
;
Gao, Yang
;
He, Shan
;
Liu, Ying
;
Lai, Luhua
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2015/11/13
PROSTAGLANDIN E-2 SYNTHASE-1
HUMAN WHOLE-BLOOD
3-DIMENSIONAL STRUCTURES
THERAPEUTIC TARGET
POTENT INHIBITORS
DUAL INHIBITORS
CYCLOOXYGENASE
BIOSYNTHESIS
INFLAMMATION
LICOFELONE
Inactivation of the E-Prostanoid 3 Receptor Attenuates the Angiotensin II Pressor Response via Decreasing Arterial Contractility
期刊论文
arteriosclerosis thrombosis and vascular biology, 2012
Chen, Lihong
;
Miao, Yifei
;
Zhang, Yahua
;
Dou, Dou
;
Liu, Limei
;
Tian, Xiaoyu
;
Yang, Guangrui
;
Pu, Dan
;
Zhang, Xiaoyan
;
Kang, Jihong
;
Gao, Yuansheng
;
Wang, Shigiang
;
Breyer, Matthew D.
;
Wang, Nanping
;
Zhu, Yi
;
Huang, Yu
;
Breyer, Richard M.
;
Guan, Youfei
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2015/11/14
angiotensin II
calcium
E-prostanoid 3
hypertension
vasoconstriction
PROSTAGLANDIN-E-RECEPTOR
SMOOTH-MUSCLE-CELLS
C-TERMINAL TAIL
BLOOD-PRESSURE
EP3 RECEPTOR
MICE LACKING
HYPERTENSION
SUBTYPE
EXPRESSION
KIDNEY
Dynamic eicosanoid responses upon different inhibitor and combination treatments on the arachidonic acid metabolic network
期刊论文
分子生物系统, 2012
He, Chong
;
Wu, Yiran
;
Lai, Yongquan
;
Cai, Zongwei
;
Liu, Ying
;
Lai, Luhua
收藏
  |  
浏览/下载:12/0
  |  
提交时间:2015/11/10
PROSTAGLANDIN E-2 SYNTHASE-1
MECHANISM-BASED INACTIVATION
HUMAN WHOLE-BLOOD
DEFICIENT MICE
POLYMORPHONUCLEAR LEUKOCYTES
5-LIPOXYGENASE 5-LOX
CELL-PROLIFERATION
TUMOR-ANGIOGENESIS
DUAL INHIBITORS
DRUG DESIGN
Microsomal prostaglandin E synthase-1 exhibits one-third-of-the-sites reactivity
期刊论文
biochemical journal, 2011
He, Shan
;
Wu, Yiran
;
Yu, Daqi
;
Lai, Luhua
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2015/11/13
drug design
enzyme mechanism
inflammation
membrane-associated proteins in eicosanoid and glutathione metabolism (MAPEG)
microsomal prostaglandin E synthase-1 (mPGES-1)
one-third-of-the-sites reactivity
UNDERSTANDING MICROSCOPIC BINDING
SITE-DIRECTED MUTAGENESIS
MOLECULAR-DYNAMICS
STRUCTURAL BASIS
FUNCTIONAL-CHARACTERIZATION
CRYSTAL-STRUCTURE
PROTEIN
SIMULATIONS
GLUTATHIONE
AMINOPEPTIDASE
Recent progress in quantitative analysis of DNA adducts of nephrotoxin aristolochic acid
期刊论文
中国科学b辑 化学英文版, 2009
Yue Hao
;
Chan Wan
;
Yu KongJie
;
Guo Lin
;
Liu Ning
;
Liu HuWei
;
Cai ZongWei
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2015/11/12
aristolochic acid
DNA adducts
quantitative analysis
short review
CHINESE HERBS NEPHROPATHY
TANDEM MASS-SPECTROMETRY
P-32 POSTLABELING ANALYSIS
PROSTAGLANDIN-H SYNTHASE
CHRONIC-RENAL-FAILURE
CYTOCHROMES P450 1A1
REDUCTIVE ACTIVATION
METABOLIC-ACTIVATION
RISK-FACTOR
RAT-KIDNEY
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