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广州生物医药与健康... [18]
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期刊论文 [18]
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2016 [2]
2015 [2]
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专题:广州生物医药与健康研究院
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GZD856, a novel potent PDGFR alpha/beta inhibitor, suppresses the growth and migration of lung cancer cells in vitro and in vivo
期刊论文
CANCER LETTERS, 2016, 卷号: 375, 期号: 1, 页码: 172-178
作者:
Song, Liyan
;
Pang, Hongwen
;
Ding, Ke
;
Yu, Rongmin
;
Zhang, Zhang
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2018/12/13
GZD856, a novel potent PDGFR alpha/beta inhibitor, suppresses the growth and migration of lung cancer cells in vitro and in vivo
期刊论文
CANCER LETTERS, 2016, 卷号: 375, 期号: 1, 页码: 172-178
Zhang, Zhang
;
Ren, Xiaomei
;
Lu, Xiaoyun
;
Wang, Deping
;
Hu, Xianjing
;
Zheng, Yi
;
Song, Liyan
;
Pang, Hongwen
;
Yu, Rongmin
;
Ding, Ke
收藏
  |  
浏览/下载:37/0
  |  
提交时间:2016/12/16
Hybrid pyrimidine alkynyls inhibit the clinically resistance related Bcr-Abl(T315I) mutant
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 17, 页码: 3458-3463
作者:
Ding, Ke
;
Pan, Xiaofeng
;
Wang, Deping
;
Zhuang, Xiaoxi
;
Luo, Jingfeng
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2018/12/13
Hybrid pyrimidine alkynyls inhibit the clinically resistance related Bcr-Abl(T315I) mutant
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 卷号: 25, 期号: 17, 页码: 3458-3463
Lu, Xiaoyun
;
Zhang, Zhang
;
Ren, Xiaomei
;
Pan, Xiaofeng
;
Wang, Deping
;
Zhuang, Xiaoxi
;
Luo, Jingfeng
;
Yu, Rongmin
;
Ding, Ke
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2016/12/16
Novel thiazole amine class tyrosine kinase inhibitors induce apoptosis in human mast cells expressing D816V KIT mutation
期刊论文
CANCER LETTERS, 2014, 卷号: 353, 期号: 1, 页码: 115-123
作者:
Wang, Deping
;
Pan, Jingxuan
;
Jin, Yanli
;
Ding, Ke
;
Shen, Mengjie
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2018/12/13
Antitumor activity of S116836, a novel tyrosine kinase inhibitor, against imatinib-resistant FIP1L1-PDGFR alpha-expressing cells
期刊论文
ONCOTARGET, 2014, 卷号: 5, 期号: 21, 页码: 10407-10420
Shen, Yingying
;
Ren, Xiaomei
;
Ding, Ke
;
Zhang, Zhang
;
Wang, Deping
;
Pan, Jingxuan
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2016/12/16
Novel thiazole amine class tyrosine kinase inhibitors induce apoptosis in human mast cells expressing D816V KIT mutation
期刊论文
CANCER LETTERS, 2014, 卷号: 353, 期号: 1, 页码: 115-123
Jin, Yanli
;
Ding, Ke
;
Wang, Deping
;
Shen, Mengjie
;
Pan, Jingxuan
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2016/12/16
Antitumor activity of S116836, a novel tyrosine kinase inhibitor, against imatinib-resistant FIP1L1-PDGFR alpha-expressing cells
期刊论文
ONCOTARGET, 2014, 卷号: 5, 期号: 21, 页码: 10407-10420
作者:
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2018/12/13
Identification of GZD824 as an Orally Bioavailable Inhibitor That Targets Phosphorylated and Nonphosphorylated Breakpoint Cluster Region-Abelson (Bcr-Abl) Kinase and Overcomes Clinically Acquired Mutation-Induced Resistance against Imatinib
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 56, 期号: 3
作者:
Wang, Deping
;
Feng, Yubing
;
Zhuang, Xiaoxi
;
Zhang, Fengxiang
;
Liu, Jianqi
收藏
  |  
浏览/下载:23/0
  |  
提交时间:2018/12/13
Identification of GZD824 as an Orally Bioavailable Inhibitor That Targets Phosphorylated and Nonphosphorylated Breakpoint Cluster Region-Abelson (Bcr-Abl) Kinase and Overcomes Clinically Acquired Mutation-Induced Resistance against Imatinib
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2013, 卷号: 56, 期号: 3
Ren, Xiaomei
;
Pan, Xiaofen
;
Zhang, Zhang
;
Wang, Deping
;
Lu, Xiaoyun
;
Li, Yupeng
;
Wen, Donghai
;
Long, Huoyou
;
Luo, Jinfeng
;
Feng, Yubing
;
Zhuang, Xiaoxi
;
Zhang, Fengxiang
;
Liu, Jianqi
;
Leng, Fang
;
Lang, Xingfen
;
Bai, Yang
;
She, Miaoqin
;
Tu, Zhengchao
;
Pan, Jingxuan
;
Ding, Ke
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2016/12/16
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