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Structural insights into ligand recognition and activation of the melanocortin-4 receptor 期刊论文
CELL RESEARCH, 2021, 页码: 13
作者:  Zhang, Huibing;  Chen, Li-Nan;  Yang, Dehua;  Mao, Chunyou;  Shen, Qingya
收藏  |  浏览/下载:34/0  |  提交时间:2021/11/04
Molecular Basis for Hormone Recognition and Activation of Corticotropin-Releasing Factor Receptors 期刊论文
MOLECULAR CELL, 2020, 卷号: 77, 期号: 3, 页码: 669-+
作者:  Ma, Shanshan;  Shen, Qingya;  Zhao, Li-Hua;  Mao, Chunyou;  Zhou, X. Edward
收藏  |  浏览/下载:16/0  |  提交时间:2020/07/01
Structure and dynamics of the active human parathyroid hormone receptor-1 期刊论文
SCIENCE, 2019, 卷号: 364, 期号: 6436, 页码: 148-+
作者:  Zhao, Li-Hua;  Ma, Shanshan;  Sutkeviciute, Ieva;  Shen, Dan-Dan;  Zhou, X. Edward
收藏  |  浏览/下载:7/0  |  提交时间:2020/07/01
Structure-based optimization of a series of selective BET inhibitors containing aniline or indoline groups 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 150, 页码: 156-175
作者:  Hu, Jianping;  Wang, Yingqing;  Li, Yanlian;  Cao, Danyan;  Xu, Lin
收藏  |  浏览/下载:34/0  |  提交时间:2019/01/08
Discovery, mechanism and metabolism studies of 2,3-difluorophenyl-linker-containing PARP1 inhibitors with enhanced in vivo efficacy for cancer therapy 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 138, 页码: 514-531
作者:  Chen, Wenhua;  Guo, Ne;  Qi, Minghui;  Dai, Haiying;  Hong, Minghuang
收藏  |  浏览/下载:30/0  |  提交时间:2019/01/08
Discovery of a series of dihydroquinoxalin-2(1H)-ones as selective BET inhibitors from a dual PLK1-BRD4 inhibitor 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 137, 页码: 176-195
作者:  Hu, Jianping;  Wang, Yingqing;  Li, Yanlian;  Xu, Lin;  Cao, Danyan
收藏  |  浏览/下载:32/0  |  提交时间:2019/01/08
Mechanism of the All-alpha to All-beta Conformational Transition of RfaH-CTD: Molecular Dynamics Simulation and Markov State Model 期刊论文
JOURNAL OF CHEMICAL THEORY AND COMPUTATION, 2014, 卷号: 10, 期号: 6, 页码: 2255-2264
作者:  Li, Shanshan;  Xiong, Bing;  Xu, Yuan;  Lu, Tao;  Luo, Xiaomin
收藏  |  浏览/下载:13/0  |  提交时间:2019/01/08
Non-Covalent Interactions with Aromatic Rings: Current Understanding and Implications for Rational Drug Design 期刊论文
CURRENT PHARMACEUTICAL DESIGN, 2013, 卷号: 19, 期号: 36, 页码: 6522-6533
作者:  Li, Shanshan;  Xu, Yuan;  Shen, Qiancheng;  Liu, Xian;  Lu, Jing
收藏  |  浏览/下载:20/0  |  提交时间:2019/01/08
In Silico Prediction of Cytochrome P450-Mediated Site of Metabolism (SOM) 期刊论文
PROTEIN AND PEPTIDE LETTERS, 2013, 卷号: 20, 期号: 3, 页码: 279-289
作者:  Liu, Xian;  Shen, Qiancheng;  Li, Jing;  Li, Shanshan;  Luo, Cheng
收藏  |  浏览/下载:8/0  |  提交时间:2019/01/08
Knowledge-Based Scoring Functions in Drug Design: 3. A Two-Dimensional Knowledge-Based Hydrogen-Bonding Potential for the Prediction of Protein-Ligand Interactions 期刊论文
JOURNAL OF CHEMICAL INFORMATION AND MODELING, 2011, 卷号: 51, 期号: 11, 页码: 2994-3004
作者:  Zheng, Mingyue;  Xiong, Bing;  Luo, Cheng;  Li, Shanshan;  Liu, Xian
收藏  |  浏览/下载:12/0  |  提交时间:2019/01/08


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