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科研机构
上海药物研究所 [9]
国家空间科学中心 [2]
新疆理化技术研究所 [1]
内容类型
期刊论文 [11]
会议论文 [1]
发表日期
2019 [12]
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Nature brings new avenues to the therapy of central nervous system diseases-An overview of possible treatments derived from natural products
期刊论文
SCIENCE CHINA-LIFE SCIENCES, 2019, 卷号: 62, 期号: 10, 页码: 1332-1367
作者:
Zhang, Junchi
;
He, Yang
;
Jiang, Xiangrui
;
Jiang, Hualiang
;
Shen, Jingshan
收藏
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浏览/下载:33/0
  |  
提交时间:2020/07/01
natural products
traditional Chinese medicine
central nervous system diseases
treatment
Metal-free quinolylation of the primary amino groups of amino acid derivatives and peptides with dihydrooxazolo[3,2-a]quinoliniums
期刊论文
GREEN CHEMISTRY, 2019, 卷号: 21, 期号: 15, 页码: 4231-4237
作者:
Liu, Peng
;
Li, Bo
;
Xi, Mengyu
;
Chen, Zhaoqiang
;
Sun, Haiguo
收藏
  |  
浏览/下载:9/0
  |  
提交时间:2020/07/01
Characterization of TPN171 metabolism in humans via ultra-performance liquid chromatography/quadrupole time-of-flight Checir for mass spectrometry
期刊论文
JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS, 2019, 卷号: 172, 页码: 302-310
作者:
Pan, Lulu
;
Guo, Shuang
;
Chen, Xiaoyan
;
Jiang, Xiangrui
;
Shen, Jingshan
收藏
  |  
浏览/下载:53/0
  |  
提交时间:2020/07/01
TPNI71
Metabolism
UPLC/Q-TOF MS
High-resolution mass spectrometry
Metabolite identification
Oxidative Aromatization of 3,4-Dihydroquinolin-2(1H)-ones to Quinolin-2(1H)-ones Using Transition-Metal-Activated Persulfate Salts
期刊论文
JOURNAL OF ORGANIC CHEMISTRY, 2019, 卷号: 84, 期号: 13, 页码: 8702-8709
作者:
Chen, Weiming
;
Sun, Changliang
;
Zhang, Yan
;
Hu, Tianwen
;
Zhu, Fuqiang
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2020/07/01
Pharmacokinetics-Driven Optimization of 4(3H)-Pyrimidinones as Phosphodiesterase Type 5 Inhibitors Leading to TPN171, a Clinical Candidate for the Treatment of Pulmonary Arterial Hypertension
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 10, 页码: 4979-4990
作者:
Wang, Zhen
;
Jiang, Xiangrui
;
Zhang, Xianglei
;
Tian, Guanghui
;
Yang, Rulei
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2020/07/01
Continuation of structure-activity relationship study of novel benzamide derivatives as potential antipsychotics
期刊论文
ARCHIV DER PHARMAZIE, 2019, 卷号: 352, 期号: 4, 页码: 13
作者:
Xu, Mingshuo
;
Guo, Shuang
;
Yang, Feipu
;
Wang, Yu
;
Wu, Chunhui
收藏
  |  
浏览/下载:43/0
  |  
提交时间:2020/07/01
5-HT1A
5-HT2A
catalepsy
D-2
PCP-induced hyperactivity
Discovery of pyrimidine nucleoside dual prodrugs and pyrazine nucleosides as novel anti-HCV agents
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2019, 卷号: 27, 期号: 5, 页码: 748-759
作者:
Guo, Shuang
;
Xu, Mingshuo
;
Guo, Qi
;
Zhu, Fuqiang
;
Jiang, Xiangrui
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2020/07/01
Nucleoside
Double prodrug
Phosphoramidate
Anti-HCV
Pyrazine
Pharmacokinetics-Driven Optimization of 4(3H)-Pyrimidinones as Phosphodiesterase Type 5 Inhibitors Leading to TPN171, a Clinical Candidate for the Treatment of Pulmonary Arterial Hypertension
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 10, 页码: 4979-4990
作者:
Wang, Z (Wang, Zhen)[ 1 ]
;
Jiang, XR (Jiang, Xiangrui)[ 1 ]
;
Zhang, XL (Zhang, Xianglei)[ 1,2 ]
;
Tian, GH (Tian, Guanghui)[ 3 ]
;
Yang, RL (Yang, Rulei)[ 3 ]
收藏
  |  
浏览/下载:137/0
  |  
提交时间:2019/06/28
Mm-wave Radar Based Micro-Deformation Monitoring for Highway and Freight Railway Bridges
会议论文
Xuzhou, PEOPLES R CHINA, JUL 21-24, 2018
作者:
Li, Yingsong
;
Shao, Zelong
;
Zhang, Xiangkun
;
Jiang, Jingshan
收藏
  |  
浏览/下载:55/0
  |  
提交时间:2019/07/10
Micro-deformation monitoring
millimeter (mm) wave radar
super-resolution and high precision
Mm-wave Radar Based Micro-Deformation Monitoring for Highway and Freight Railway Bridges
期刊论文
APPLIED COMPUTATIONAL ELECTROMAGNETICS SOCIETY JOURNAL, 2019, 卷号: 34, 期号: 3, 页码: 457-462
作者:
Li, Yingsong
;
Shao, Zelong
;
Zhang, Xiangkun
;
Jiang, Jingshan
收藏
  |  
浏览/下载:57/0
  |  
提交时间:2019/07/10
Micro-deformation Monitoring
Millimeter (Mm) Wave Radar
Super-resolution And High Precision
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