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科研机构
上海药物研究所 [26]
内容类型
期刊论文 [26]
发表日期
2018 [1]
2016 [1]
2014 [1]
2013 [1]
2012 [1]
2011 [1]
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Characteristics of hERG and hNav1.5 channel blockade by sulcardine sulfate, a novel anti-arrhythmic compound
期刊论文
European journal of pharmacology, 2018, 卷号: 844, 页码: 130-138
作者:
Chen, Weihai
;
Gan, Lu
;
Wang, Yiping
收藏
  |  
浏览/下载:18/0
  |  
提交时间:2019/01/08
Propofol inhibits hERG K+ channels and enhances the inhibition effects on its mutations in HEK293 cells
期刊论文
EUROPEAN JOURNAL OF PHARMACOLOGY, 2016, 卷号: 791, 页码: 168-178
作者:
Han, Sheng-Na
;
Jing, Ying
;
Yang, Lin-Lin
;
Zhang, Zhao
;
Zhang, Li-Rong
收藏
  |  
浏览/下载:42/0
  |  
提交时间:2019/01/08
Propofol
QT prolongation
Human ether-a-go-go-related gene (hERG)
Protein trafficking
Gene mutation
Development of Mechanostimulated Patch-Clamp System for Cellular Physiological Study
期刊论文
IEEE-ASME TRANSACTIONS ON MECHATRONICS, 2014, 卷号: 19, 期号: 4, 页码: 1138-1147
作者:
Zhang, Changlin
;
Li, Peng
;
Liu, Lianqing
;
Wang, Yuechao
;
Gao, Zhaobing
收藏
  |  
浏览/下载:30/0
  |  
提交时间:2019/01/08
Atomic force microscope (AFM)
mechanosensitive (MS) ion channel
planar patch clamp
Properties and Molecular Determinants of the Natural Flavone Acacetin for Blocking hKv4.3 Channels
期刊论文
PLOS ONE, 2013, 卷号: 8, 期号: 3
作者:
Wu, Hui-Jun
;
Sun, Hai-Ying
;
Wu, Wei
;
Zhang, Yan-Hui
;
Qin, Guo-Wei
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2019/01/08
Comparison of the effects of DC031050, a class III antiarrhythmic agent, on hERG channel and three neuronal potassium channels
期刊论文
ACTA PHARMACOLOGICA SINICA, 2012, 卷号: 33, 期号: 6, 页码: 728-736
作者:
Li, Ping
;
Sun, Hai-feng
;
Zhou, Ping-zheng
;
Ma, Chao-ying
;
Hu, Guo-yuan
收藏
  |  
浏览/下载:39/0
  |  
提交时间:2019/01/08
dofetilide
DC031050
class III antiarrhythmic agent
hERG
KCNQ
Kv1.2
delayed rectifier potassium current
Acacetin causes a frequency- and use-dependent blockade of hKv1.5 channels by binding to the S6 domain
期刊论文
JOURNAL OF MOLECULAR AND CELLULAR CARDIOLOGY, 2011, 卷号: 51, 期号: 6, 页码: 966-973
作者:
Wu, Hui-Jun
;
Wu, Wei
;
Sun, Hai-Ying
;
Qin, Guo-Wei
;
Wang, Hong-Bing
收藏
  |  
浏览/下载:17/0
  |  
提交时间:2019/01/08
Acacetin
hKv1.5
Tonic blockade
Open channel blockade
Rate-dependent blockade
Cellular electrophysiological effects of changrolin in isolated rat cardiac myocytes
期刊论文
EUROPEAN JOURNAL OF PHARMACOLOGY, 2010, 卷号: 647, 期号: 1-3, 页码: 139-146
作者:
Chen, Wei-hai
;
Yang, Ding
;
Wang, Wen-yi
;
Zhang, Jie
;
Wang, Yi-ping
收藏
  |  
浏览/下载:14/0
  |  
提交时间:2019/01/08
Changrolin
Whole-cell patch-clamp
Na+ channels
K+ channels
Ca2+ channels
State-dependent blockade of human ether-a-go-go-related gene (hERG) K+ channels by changrolin in stably transfected HEK293 cells
期刊论文
ACTA PHARMACOLOGICA SINICA, 2010, 卷号: 31, 期号: 8, 页码: 915-922
作者:
Chen, Wei-hai
;
Wang, Wen-yi
;
Zhang, Jie
;
Yang, Ding
;
Wang, Yi-ping
收藏
  |  
浏览/下载:13/0
  |  
提交时间:2019/01/08
changrolin
human ether-a-go-go-related gene
torsades de pointes
whole-cell patch-clamp
anti-arrhythmic agent
Magnesium lithospermate B dilates mesenteric arteries by activating BKCa currents and contracts arteries by inhibiting K-V currents
期刊论文
ACTA PHARMACOLOGICA SINICA, 2010, 卷号: 31, 期号: 6, 页码: 665-670
作者:
Zhang, Hai-fei
;
Chen, Xue-qing
;
Hu, Guo-yuan
;
Wang, Yi-ping
收藏
  |  
浏览/下载:16/0
  |  
提交时间:2019/01/08
magnesium lithospermate B
big-conductance Ca2+-activated K+ channels
mesenteric artery
endothelium
State-dependent blockade of human ether-a-go-go-related gene (hERG) K~+ channels by changrolin in stably transfected HEK293 cells
期刊论文
Acta Pharmacologica Sinica, 2010, 卷号: 31, 期号: 8, 页码: 915
作者:
Chen Weihai
;
Wang Wenyi
;
Zhang Jie
;
Yang Ding
;
Wang Yiping
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2020/07/01
TORSADES-DE-POINTES
POTASSIUM CHANNELS
PROLONGATION
DERIVATIVES
BINDING
DRUGS
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