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Discovery of an Inhibitor for the TREK-1 Channel Targeting an Intermediate Transition State of Channel Gating 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 19, 页码: 10972-10983
作者:  Ma, Yuqin;  Luo, Qichao;  Fu, Jie;  Che, Yanxin;  Guo, Fei
收藏  |  浏览/下载:11/0  |  提交时间:2021/05/24
Antiepileptic geissoschizine methyl ether is an inhibitor of multiple neuronal channels 期刊论文
ACTA PHARMACOLOGICA SINICA, 2020, 页码: 9
作者:  Xie, Zhu-qing;  Tian, Xiao-ting;  Zheng, Yue-ming;  Zhan, Li;  Chen, Xue-qin
收藏  |  浏览/下载:23/0  |  提交时间:2020/07/01
Selective activation of TWIK-related acid-sensitive K+ 3 subunit-containing channels is analgesic in rodent models 期刊论文
SCIENCE TRANSLATIONAL MEDICINE, 2019, 卷号: 11, 期号: 519, 页码: 12
作者:  Liao, Ping;  Qiu, Yunguang;  Mo, Yiqing;  Fu, Jie;  Song, Zhenpeng
收藏  |  浏览/下载:30/0  |  提交时间:2020/07/01
A Statistical Thermodynamic Model for Ligands Interacting With Ion Channels: Theoretical Model and Experimental Validation of the KCNQ2 Channel 期刊论文
FRONTIERS IN PHARMACOLOGY, 2018, 卷号: 9
作者:  Bai, Fang;  Pi, Xiaoping;  Li, Ping;  Zhou, Pingzheng;  Yang, Huaiyu
收藏  |  浏览/下载:29/0  |  提交时间:2019/01/08
Enhanced stability of vitamin A palmitate microencapsulated by gamma-cyclodextrin metal-organic frameworks 期刊论文
JOURNAL OF MICROENCAPSULATION, 2018, 卷号: 35, 期号: 3, 页码: 249-258
作者:  Zhang, Guoqing;  Meng, Fanyue;  Guo, Zhen;  Guo, Tao;  Peng, Hui
收藏  |  浏览/下载:20/0  |  提交时间:2019/01/08
An allosteric ligand-binding site in the extracellular cap of K2P channels 期刊论文
NATURE COMMUNICATIONS, 2017, 卷号: 8
作者:  Luo, Qichao;  Chen, Liping;  Cheng, Xi;  Ma, Yuqin;  Li, Xiaona
收藏  |  浏览/下载:17/0  |  提交时间:2019/01/08
Grafting voltage and pharmacological sensitivity in potassium channels 期刊论文
CELL RESEARCH, 2016, 卷号: 26, 期号: 8, 页码: 935-945
作者:  Lan, Xi;  Fan, Chunyan;  Ji, Wei;  Tian, Fuyun;  Xu, Tao
收藏  |  浏览/下载:14/0  |  提交时间:2019/01/08
SP6616 as a new Kv2.1 channel inhibitor efficiently promotes beta-cell survival involving both PKC/Erk1/2 and CaM/PI3K/Akt signaling pathways 期刊论文
CELL DEATH & DISEASE, 2016, 卷号: 7
作者:  Zhou, T. T.;  Quan, L. L.;  Chen, L. P.;  Du, T.;  Sun, K. X.
收藏  |  浏览/下载:25/0  |  提交时间:2019/01/08
Novel analogues of diterpenoid alkaloids from ring distortion of talatisamine, a potassium ion channel blocker 期刊论文
TETRAHEDRON, 2016, 卷号: 72, 期号: 10, 页码: 1357-1363
作者:  Tang, Hua;  Chen, Qi-Feng;  Liu, Xiao-Yu;  Zhang, Hua;  Chen, Dong-Lin
收藏  |  浏览/下载:13/0  |  提交时间:2019/01/08
Computer-Aided Drug Discovery and Design Targeting Ion Channels 期刊论文
CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2016, 卷号: 16, 期号: 16, 页码: 1819-1829
作者:  Zhang, Qiansen;  Gao, Zhaobing;  Yang, Huaiyu
收藏  |  浏览/下载:36/0  |  提交时间:2019/01/08


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