CORC

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Synthesis and PTP1B/TCPTP Inhibitory Activity Evaluation of Novel 2,5-Disubstituted-1,3,4-thiadiazolamide Derivatives Containing Carbazole/Benzimidazole Moity 期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2019, 卷号: 39, 期号: 9, 页码: 2599-2608
作者:  Li Yingjun;  Zhao Yue;  Jin Kun;  Gao Lixin;  Sheng Li
收藏  |  浏览/下载:34/0  |  提交时间:2020/07/01
Discovery of novel high potent and cellular active ADC type PTP1B inhibitors with selectivity over TC-PTP via modification interacting with C site 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2018, 卷号: 144, 页码: 692-700
作者:  Du, Yongli;  Zhang, Yanhui;  Ling, Hao;  Li, Qunyi;  Shen, Jingkang
收藏  |  浏览/下载:20/0  |  提交时间:2019/01/08
Conformation and dynamics of the C-terminal region in human phosphoglycerate mutase 1 期刊论文
ACTA PHARMACOLOGICA SINICA, 2017, 卷号: 38, 期号: 12, 页码: 1673-1682
作者:  Liu, Shi-en;  Hu, Jun-chi;  Zhang, Hao;  Xu, Pan;  Wan, Wei
收藏  |  浏览/下载:19/0  |  提交时间:2019/01/08
Pyrazolopyrimidines as Potent Stimulators for Transient Receptor Potential Canonical 3/6/7 Channels 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 11, 页码: 4680-4692
作者:  Qu, Chunrong;  Ding, Mingmin;  Zhu, Yingmin;  Lu, Yungang;  Du, Juan
收藏  |  浏览/下载:89/0  |  提交时间:2019/01/08
Discovery of di-indolinone as a novel scaffold for protein tyrosine phosphatase 1B inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 卷号: 22, 期号: 24, 页码: 7440-7443
作者:  Dai, Hou-ling;  Gao, Li-xin;  Yang, Ying;  Li, Jing-ya;  Cheng, Jia-gao
收藏  |  浏览/下载:18/0  |  提交时间:2019/01/08
Facile fabrication of promising protein tyrosine phosphatase (PTP) inhibitor entities based on 'clicked' serine/threonine-monosaccharide hybrids 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2011, 卷号: 19, 期号: 13, 页码: 3892-3900
作者:  He, Xiao-Peng;  Deng, Qiong;  Gao, Li-Xin;  Li, Cui;  Zhang, Wei
收藏  |  浏览/下载:17/0  |  提交时间:2019/01/08
Monosaccharide as a Central Scaffold Toward the Construction of Salicylate-Based Bidentate PTP1B Inhibitors via Click Chemistry 期刊论文
BULLETIN OF THE KOREAN CHEMICAL SOCIETY, 2011, 卷号: 32, 期号: 3, 页码: 1000-1006
作者:  Tang, Yan-Hui;  Hu, Min;  He, Xiao-Peng;  Fahnbulleh, Sando;  Li, Cui
收藏  |  浏览/下载:8/0  |  提交时间:2019/01/08
Triazole-linked Benzylated Glucosyl, Galactosyl, and Mannosyl Monomers and Dimers as Novel Sugar Scaffold-based PTP1B Inhibitors 期刊论文
CHEMISTRY LETTERS, 2010, 卷号: 39, 期号: 12, 页码: 1261-1263
作者:  Zhang, Yin Jie;  He, Xiao-Peng;  Li, Cui;  Li, Zhen;  Shi, De-Tai
收藏  |  浏览/下载:8/0  |  提交时间:2019/01/08
Microwave-Accelerated Click Chemistry: Expeditious Synthesis of Novel Triazole-linked Salicylic beta-D-O-Glycosides with PTP1B Inhibitory Activity 期刊论文
BULLETIN OF THE KOREAN CHEMICAL SOCIETY, 2010, 卷号: 31, 期号: 11, 页码: 3359-3365
作者:  Yang, Jin-Wei;  Li, Cui;  He, Xiao-Peng;  Zhao, Hong;  Gao, Li-Xin
收藏  |  浏览/下载:12/0  |  提交时间:2019/01/08
Synthesis and LAR inhibition of 7-alkoxy analogues of illudalic acid 期刊论文
Yao xue xue bao = Acta pharmaceutica Sinica, 2010, 卷号: 45, 期号: 11, 页码: 1385-97
作者:  Ling, Qing;  Zhou, Yue-Yang;  Cai, Zheng-Liang;  Zhang, Ya-Hui;  Xiong, Bing
收藏  |  浏览/下载:5/0  |  提交时间:2019/01/08


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