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Natural Product Albiziabioside A Conjugated with Pyruvate Dehydrogenase Kinase Inhibitor Dichloroacetate To Induce Apoptosis-Ferroptosis-M2-TAMs Polarization for Combined Cancer Therapy 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2019, 卷号: 62, 期号: 19, 页码: 8760-8772
作者:  Wei, Gaofei;  Sung, Jiahong;  Luan, Weijing;  Hou, Zhuang;  Wang, Shuai
收藏  |  浏览/下载:18/0  |  提交时间:2020/07/01
Development of the First Generation of Disulfide-Based Subtype Selective and Potent Covalent Pyruvate Dehydrogenase Kinase 1 (PDK1) Inhibitors 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 6, 页码: 2227-2244
作者:  Liu, Yifu;  Xie, Zuoquan;  Zhao, Dan;  Zhu, Jin;  Mao, Fei
收藏  |  浏览/下载:22/0  |  提交时间:2019/01/08
JX06 Selectively Inhibits Pyruvate Dehydrogenase Kinase PDK1 by a Covalent Cysteine Modification 期刊论文
CANCER RESEARCH, 2015, 卷号: 75, 期号: 22, 页码: 4923-4936
作者:  Sun, Wenyi;  Xie, Zuoquan;  Liu, Yifu;  Zhao, Dan;  Wu, Zhixiang
收藏  |  浏览/下载:29/0  |  提交时间:2019/01/08
Design, synthesis and anticancer activity of diam(m)ine platinum(II) complexes bearing a small-molecular cell apoptosis inducer dichloroacetate 期刊论文
JOURNAL OF INORGANIC BIOCHEMISTRY, 2015, 卷号: 146, 页码: 14-18
作者:  Liu, Weiping;  Jiang, Jing;  Xu, Yongping;  Hou, Shuqian;  Sun, Liping
收藏  |  浏览/下载:17/0  |  提交时间:2019/01/08
Discovery and Optimization of 4,5-Diarylisoxazoles as Potent Dual Inhibitors of Pyruvate Dehydrogenase Kinase and Heat Shock Protein 90 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2014, 卷号: 57, 期号: 23, 页码: 9832-9843
作者:  Meng, Tao;  Zhang, Dadong;  Xie, Zuoquan;  Yu, Ting;  Wu, Shuchao
收藏  |  浏览/下载:8/0  |  提交时间:2019/01/08
Synthesis, anticancer activity and toxicity of a water-soluble 4S,5S-derivative of heptaplatin, cis-{Pt(II)[(4S,5S)-4,5-bis(aminomethyl)-2-isopropyl-1,3-dioxolane].(3-hydroxyl-cyclobutane-1,1-dicarboxylate)} 期刊论文
JOURNAL OF INORGANIC BIOCHEMISTRY, 2014, 卷号: 140, 页码: 126-130
作者:  Liu, Weiping;  Jiang, Jing;  Xie, Chengying;  Hou, Shuqian;  Quan, Haitian
收藏  |  浏览/下载:15/0  |  提交时间:2019/01/08


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