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科研机构
上海药物研究所 [62]
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期刊论文 [62]
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2021 [4]
2020 [4]
2019 [4]
2018 [7]
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Theoretical study and application of 2-phenyl-1,3,4-thiadiazole derivatives with optical and inhibitory activity against SHP1
期刊论文
PHYSICAL CHEMISTRY CHEMICAL PHYSICS, 2021, 页码: 14
作者:
Zhang, Chun
;
Sun, Yi-Tao
;
Gao, Li-Xin
;
Feng, Bo
;
Yan, Xue
收藏
  |  
浏览/下载:21/0
  |  
提交时间:2022/01/18
Synthesis and Protein Tyrosine Phosphatase 1B (PTP1B) Inhibitory Activity Evaluation of Novel N-Acylhydrazone Derivatives Containing Carbazole and Aromatic Ring/Aromatic Fused Heterocycle
期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 41, 期号: 9, 页码: 3593-3607
作者:
Li Yingjun
;
Lin Ledi
;
Liu Jihong
;
Gao Lixin
;
Sheng Li
收藏
  |  
浏览/下载:19/0
  |  
提交时间:2021/12/01
PTP1B inhibitor
carbazole
N-actylhydrazone
synthesis
molecular docking
Synthesis and Protein Tyrosine Phosphatase 1B (PTP1B) Inhibitory Activity Evaluation of Novel Arylaminoacetylhydrazone Derivatives Containing Carbazole Moiety
期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2021, 卷号: 41, 期号: 8, 页码: 3157-3170
作者:
Li Yingjun
;
Lin Ledi
;
Jin Kun
;
Gao Lixin
;
Sheng Li
收藏
  |  
浏览/下载:22/0
  |  
提交时间:2021/11/04
protein tyrosine phosphatase 1B (PTP1B) inhibitor
carbazole
arylaminoacetylhydrazone
synthesis
molecular docking
Synthesis of 2-ethoxycarbonylthieno[2,3-b]quinolines in biomass-derived solvent gamma-valerolactone and their biological evaluation against protein tyrosine phosphatase 1B
期刊论文
RSC ADVANCES, 2021, 卷号: 11, 期号: 6, 页码: 3216-3220
作者:
Mu, Xu-Yang
;
Wang, Zhi-Jia
;
Feng, Bo
;
Xu, Lei
;
Gao, Li-Xin
收藏
  |  
浏览/下载:15/0
  |  
提交时间:2021/05/24
Sweroside promotes osteoblastic differentiation and mineralization via interaction of membrane estrogen receptor-alpha and GPR30 mediated p38 signalling pathway on MC3T3-E1 cells
期刊论文
PHYTOMEDICINE, 2020, 卷号: 68, 页码: 12
作者:
Wu, Qing-Chang
;
Tang, Xi-Yang
;
Dai, Zi-Qin
;
Dai, Yi
;
Xiao, Hui-Hui
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2020/07/01
Sweroside
Differentiation and mineralization
Membrane estrogen receptor-alpha
GPR30
P38 signaling pathway
MC3T3-E1 cells
Synthesis and Protein Tyrosine Phosphatase 1B (PTP1B) Inhibitory Activity Evaluation of Novel Carbazole-Based Carbohydrazone Derivatives
期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2020, 卷号: 40, 期号: 2, 页码: 478-488
作者:
Li, Yingjun
;
Liu, Xuejie
;
Liu, Jihong
;
Gao, Lixin
;
Jin, Kun
收藏
  |  
浏览/下载:44/0
  |  
提交时间:2020/07/01
carbohydrazone
carbazole
synthesis
PTP1B inhibitor
molecular docking
DFT calculations
Spirobiflavonoid stereoisomers from the endangered conifer Glyptostrobus pensilis and their protein tyrosine phosphatase 1B inhibitory activity
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2020, 卷号: 30, 期号: 4, 页码: 4
作者:
Xiong, Juan
;
Hu, Chang-Ling
;
Wang, Pei-Pei
;
Gao, Ding-Ding
;
Huang, Fang
收藏
  |  
浏览/下载:45/0
  |  
提交时间:2020/07/01
Glyptostrobus pensilis
Cupressaceae
Endangered conifer
Spirobiflavonoids
PTP1B inhibition
Phytochemical and biological studies on rare and endangered plants endemic to China. Part XIV. Structurally diverse terpenoids from the twigs and needles of the endangered plant Picea brachytyla
期刊论文
PHYTOCHEMISTRY, 2020, 卷号: 169, 页码: 11
作者:
Jiang, Wei
;
Xiong, Juan
;
Zang, Yi
;
Li, Junmin
;
Osman, Ezzat E. A.
收藏
  |  
浏览/下载:84/0
  |  
提交时间:2020/07/01
Picea brachytyla (Franch.) E.Pritz.
Pinaceae
Endangered plant
Terpenoids
Brachytylins
ATP citrate lyase (ACL)
SHP2 tyrosine phosphatase
Synthesis and PTP1B/TCPTP Inhibitory Activity Evaluation of Novel 2,5-Disubstituted-1,3,4-thiadiazolamide Derivatives Containing Carbazole/Benzimidazole Moity
期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2019, 卷号: 39, 期号: 9, 页码: 2599-2608
作者:
Li Yingjun
;
Zhao Yue
;
Jin Kun
;
Gao Lixin
;
Sheng Li
收藏
  |  
浏览/下载:35/0
  |  
提交时间:2020/07/01
1,3,4-thiadiazolamide
carbazole
benzimidazole
synthesis
PTP1B inhibitor
molecular docking
density functional theory (DFT) study
Synthesis and PTP1B Inhibitory Activity of Novel Chalcone Derivatives Bearing 1H-Benzo[d]imidazol or 1H-Benzo[d][1,2,3]triazol Moieties
期刊论文
CHINESE JOURNAL OF ORGANIC CHEMISTRY, 2019, 卷号: 39, 期号: 4, 页码: 1029-1036
作者:
Fu Yang
;
Sheng Li
;
Gao Lixin
;
Li Jia
;
Sun Liangpeng
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2020/07/01
PTP1B inhibitor
1H-benzo[d]imidazol
1H-benzo[d][1,2,3]triazol
chalcone
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