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Optimization of piperidine constructed peptidyl derivatives as proteasome inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2021, 卷号: 29, 页码: 14
作者:  Zhao, Yanmei;  Xu, Lei;  Zhang, Jiankang;  Zhang, Mengmeng;  Lu, Jingyi
收藏  |  浏览/下载:21/0  |  提交时间:2021/05/24
Peptidyl-Lys metalloendopeptidase (Lys-N) purified from dry fruit of Grifola frondosa demonstrates "mirror"digestion property with lysyl endopeptidase (Lys-C) 期刊论文
RAPID COMMUNICATIONS IN MASS SPECTROMETRY, 2020, 卷号: 34, 期号: 2, 页码: 11
作者:  Zhao, Mingzhi;  Hao, Bingbing;  Li, Honghao;  Cai, Man;  Xie, Jingjing
收藏  |  浏览/下载:18/0  |  提交时间:2020/07/01
Exploration of novel piperazine or piperidine constructed non-covalent peptidyl derivatives as proteasome inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 126, 页码: 1056-1070
作者:  Zhuang, Rangxiao;  Gao, Lixin;  Lv, Xiaoqing;  Xi, Jianjun;  Sheng, Li
收藏  |  浏览/下载:21/0  |  提交时间:2019/01/08
Design, synthesis and biological evaluation of novel non-covalent piperidine-containing peptidyl proteasome inhibitors 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2016, 卷号: 24, 期号: 23, 页码: 6206-6214
作者:  Zhang, Jiankang;  Gao, Lixin;  Xi, Jianjun;  Sheng, Li;  Zhao, Yanmei
收藏  |  浏览/下载:51/0  |  提交时间:2019/01/08
Identification and biochemical characterization of DC07090 as a novel potent small molecule inhibitor against human enterovirus 71 3C protease by structure-based virtual screening 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2016, 卷号: 124, 页码: 981-991
作者:  Ma, Guang-Hui;  Ye, Yan;  Zhang, Dan;  Xu, Xin;  Si, Pei
收藏  |  浏览/下载:29/0  |  提交时间:2019/01/08
Design, Synthesis and Biological Evaluation of Peptidyl Epoxyketone Proteasome Inhibitors Composed of beta-amino Acids 期刊论文
CHEMICAL BIOLOGY & DRUG DESIGN, 2014, 卷号: 84, 期号: 5, 页码: 497-504
作者:  Zhang, Jiankang;  Han, Mengmeng;  Ma, Xiaodong;  Xu, Lei;  Cao, Jiayi
收藏  |  浏览/下载:15/0  |  提交时间:2019/01/08
Solution Structural Analysis of the Single-Domain Parvulin TbPin1 期刊论文
PLOS ONE, 2012, 卷号: 7, 期号: 8
作者:  Sun, Lifang;  Wu, Xueji;  Peng, Yu;  Goh, Jian Yuan;  Liou, Yih-Cherng
收藏  |  浏览/下载:14/0  |  提交时间:2019/01/08
Structure-based identification of small molecule compounds targeting cell cyclophilin A with anti-HIV-1 activity 期刊论文
EUROPEAN JOURNAL OF PHARMACOLOGY, 2007, 卷号: 565, 期号: 1-3, 页码: 54-59
作者:  Chen, Shuai;  Zhao, Xuemei;  Tan, Jinzhi;  Lu, Hong;  Qi, Zhi
收藏  |  浏览/下载:14/0  |  提交时间:2019/01/08
One novel quinoxaline derivative as a potent human cyclophilin A inhibitor shows highly inhibitory activity against mouse spleen cell proliferation 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2006, 卷号: 14, 期号: 16, 页码: 5527-5534
作者:  Li, Jian;  Chen, Jing;  Zhang, Li;  Wang, Feng;  Gui, Chunshan
收藏  |  浏览/下载:14/0  |  提交时间:2019/01/08
Discovering novel chemical inhibitors of human cyclophilin A: Virtual screening, synthesis, and bioassay 期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2006, 卷号: 14, 期号: 7, 页码: 2209-2224
作者:  Li, J;  Chen, J;  Gui, CS;  Zhang, L;  Qin, Y
收藏  |  浏览/下载:14/0  |  提交时间:2019/01/08


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