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科研机构
北京大学 [187]
内容类型
期刊论文 [167]
其他 [20]
发表日期
2017 [12]
2016 [22]
2015 [17]
2014 [26]
2013 [25]
2012 [17]
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共187条,第1-10条
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专题:北京大学
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Increased GSNOR Expression during Aging Impairs Cognitive Function and Decreases S-Nitrosation of CaMKII alpha
期刊论文
JOURNAL OF NEUROSCIENCE, 2017
Zhang, Yuying
;
Wu, Kaiyuan
;
Su, Wenting
;
Zhang, Deng-Feng
;
Wang, Ping
;
Qiao, Xinhua
;
Yao, Qin
;
Yuan, Zengqiang
;
Yao, Yong-Gang
;
Liu, Guanghui
;
Zhang, Chen
;
Liu, Limin
;
Chen, Chang
收藏
  |  
浏览/下载:11/0
  |  
提交时间:2017/12/03
age-related cognitive impairment
CaMKII alpha
nitric oxide
S-nitrosation modification
S-nitrosoglutathione reductase
LONG-TERM POTENTIATION
CENTRAL-NERVOUS-SYSTEM
NITRIC-OXIDE SYNTHASE
MORRIS WATER MAZE
NITROSOGLUTATHIONE REDUCTASE
SPATIAL MEMORY
NEURODEGENERATIVE DISEASES
SYNAPTIC PLASTICITY
DENDRITIC SPINES
GENE-EXPRESSION
Synthesis and evaluation of osimertinib derivatives as potent EGFR inhibitors
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2017
Gao, Hongying
;
Yang, Zimo
;
Yang, Xinglin
;
Rao, Yu
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2017/12/03
Osimertinib
N-Oxide metabolites
Fluoride
Non-small cell lung cancer
Epidermal growth factor receptor-tyrosine kinase inhibitors
CELL LUNG-CANCER
FACTOR RECEPTOR EGFR
MEDICINAL CHEMISTRY
TARGETED THERAPY
DRUG DISCOVERY
RESISTANCE
FLUORINE
MUTATIONS
MUTANT
PHARMACOKINETICS
Covalent Probe Finds Carboxylic Acid
期刊论文
CELL CHEMICAL BIOLOGY, 2017
Jones, Alexander
;
Zhang, Xiaoyun
;
Lei, Xiaoguang
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2017/12/03
NF-kappa B signaling and cell-fate decision induced by a fast-dissociating tumor necrosis factor mutant
期刊论文
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS, 2017
Zhang, Xiaoling
;
Yin, Ning
;
Guo, Annan
;
Zhang, Qi
;
Zhang, Yalei
;
Xu, Youjun
;
Liu, Hongbo
;
Tang, Bo
;
Lai, Luhua
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2017/12/03
NF-kappa B signaling dynamics
TNF
Receptor-ligand binding kinetics
Gene expression
Biased activation
Apoptosis
GENE-EXPRESSION
DYNAMICS
SPECIFICITY
DETERMINES
KINETICS
ALPHA
TNF
Biomimetically inspired asymmetric total synthesis of (+)-19-dehydroxyl arisandilactone A
期刊论文
Nature Communications, 2017
Han, Yi-Xin
;
Jiang, Yan-Long
;
Li, Yong
;
Yu, Hai-Xin
;
Tong, Bing-Qi
;
Niu, Zhe
;
Zhou, Shi-Jie
;
Liu, Song
;
Lan, Yu
;
Chen, Jia-Hua
;
Yang, Zhen
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2017/12/03
SCHISANDRA-ARISANENSIS
TRITERPENOIDS
ESTERS
FRUITS
FAMILY
Discovery of a Highly Potent, Selective, and Metabolically Stable Inhibitor of Receptor-Interacting Protein 1 (RIP1) for the Treatment of Systemic Inflammatory Response Syndrome
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017
Ren, Yan
;
Su, Yaning
;
Sun, Liming
;
He, Sudan
;
Meng, Lingjun
;
Liao, Daohong
;
Liu, Xiao
;
Ma, Yongfen
;
Liu, Chunyan
;
Li, Sisi
;
Ruan, Hanying
;
Lei, Xiaoguang
;
Wang, Xiaodong
;
Zhang, Zhiyuan
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2017/12/03
EXPERIMENTAL DISEASE-MODELS
CELL-DEATH
KINASE INHIBITORS
INDUCED SHOCK
NECROPTOSIS
NECROSIS
NECROSTATIN-1
SPECIFICITY
INJURY
ALPHA
PDTCM: a systems pharmacology platform of traditional Chinese medicine for psoriasis
期刊论文
ANNALS OF MEDICINE, 2017
Wang, Dongmei
;
Gu, Jiangyong
;
Zhu, Wei
;
Luo, Fang
;
Chen, Lirong
;
Xu, Xiaojie
;
Lu, Chuanjian
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2017/12/03
High throughput virtual screening
psoriasis
systems pharmacology
target prediction
traditional Chinese medicine
DRUG DISCOVERY
NATURAL-PRODUCTS
CHEMICAL SPACE
EVOLVING ROLE
PSORI-CM01
VULGARIS
DATABASE
THERAPY
FORMULA
PATHOGENESIS
Mechanistic Study of SmI2-Mediated Reformatsky Reaction for Macrolactam Formation Using a Cyclopropyl Group as a Probe
期刊论文
ISRAEL JOURNAL OF CHEMISTRY, 2017
Yang, Shouliang
;
Xi, Yumeng
;
Chen, Jiahua
;
Yang, Zhen
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2017/12/03
bromine
carbon
macrolactam formation
mechanistic study
SmI2-mediated Reformatsky reaction
ORGANIC-SYNTHESIS
TETRAPETALONE-A
STREPTOMYCES SP
SAMARIUM(II) IODIDE
NATURAL-PRODUCTS
DRUG DISCOVERY
RING
HYDROXYLATION
LANTHANIDES
REDUCTION
Small molecule enabled chemical biology and drug discovery Preface
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY, 2017
Lei, Xiaoguang
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2017/12/03
Rational Design of Selective Allosteric Inhibitors of PHGDH and Serine Synthesis with Anti-tumor Activity
期刊论文
CELL CHEMICAL BIOLOGY, 2017
Wang, Qian
;
Liberti, Maria V.
;
Liu, Pei
;
Deng, Xiaobing
;
Liu, Ying
;
Locasale, Jason W.
;
Lai, Luhua
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2017/12/03
PHOSPHOGLYCERATE DEHYDROGENASE
CANCER METABOLISM
SYNTHESIS PATHWAY
ACCURATE DOCKING
BINDING-SITES
DRUG DESIGN
BIOSYNTHESIS
DISCOVERY
CELLS
COMBINATION
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