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科研机构
北京大学 [19]
内容类型
期刊论文 [18]
其他 [1]
发表日期
2017 [2]
2016 [1]
2015 [1]
2014 [5]
2013 [2]
2012 [1]
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专题:北京大学
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Rational Design of Selective Allosteric Inhibitors of PHGDH and Serine Synthesis with Anti-tumor Activity
期刊论文
CELL CHEMICAL BIOLOGY, 2017
Wang, Qian
;
Liberti, Maria V.
;
Liu, Pei
;
Deng, Xiaobing
;
Liu, Ying
;
Locasale, Jason W.
;
Lai, Luhua
收藏
  |  
浏览/下载:1/0
  |  
提交时间:2017/12/03
PHOSPHOGLYCERATE DEHYDROGENASE
CANCER METABOLISM
SYNTHESIS PATHWAY
ACCURATE DOCKING
BINDING-SITES
DRUG DESIGN
BIOSYNTHESIS
DISCOVERY
CELLS
COMBINATION
Functional Built-In Template Directed Siliceous Fluorescent Supramolecular Vesicles as Diagnostics
期刊论文
ACS APPLIED MATERIALS & INTERFACES, 2017
Li, Jie
;
Liu, Kaerdun
;
Chen, Hengyu
;
Li, Ruoyan
;
Drechsler, Markus
;
Bai, Fan
;
Huang, Jianbin
;
Tang, Ben Zhong
;
Yan, Yun
收藏
  |  
浏览/下载:5/0
  |  
提交时间:2017/12/03
hybrid self-assembly
aggregation-induced emission
template
fluorescent vesicles
precision medicine
AGGREGATION-INDUCED EMISSION
RESONANCE ENERGY-TRANSFER
MESOPOROUS SILICA
DRUG-DELIVERY
COLORIMETRIC ASSAY
THERANOSTIC NANOMEDICINE
CANCER-THERAPY
AIE LUMINOGEN
FOLIC-ACID
NANOPARTICLES
New Mechanistic Insights on the Selectivity of Transition-Metal-Catalyzed Organic Reactions: The Role of Computational Chemistry
期刊论文
ACCOUNTS OF CHEMICAL RESEARCH, 2016
Zhang, Xinhao
;
Chung, Lung Wa
;
Wu, Yun-Dong
收藏
  |  
浏览/下载:6/0
  |  
提交时间:2017/12/03
C-H ACTIVATION
O BOND FORMATION
ASYMMETRIC HYDROGENATION
ALKYNE HYDROSILYLATION
RUTHENIUM COMPLEXES
INTERNAL ALKYNES
LIGAND
ARYLATION
ENANTIOSELECTION
AMINATION
Meclofenamic acid selectively inhibits FTO demethylation of m(6)A over ALKBH5
期刊论文
核酸研究, 2015
Huang, Yue
;
Yan, Jingli
;
Li, Qi
;
Li, Jiafei
;
Gong, Shouzhe
;
Zhou, Hu
;
Gan, Jianhua
;
Jiang, Hualiang
;
Jia, Gui-Fang
;
Luo, Cheng
;
Yang, Cai-Guang
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2015/11/15
PROMOTE PROTEIN STABILITY
OBESITY-ASSOCIATED FTO
OXIDATIVE DEMETHYLATION
CRYSTAL-STRUCTURES
RNA DEMETHYLASE
ALKYLATION DAMAGE
ESCHERICHIA-COLI
MESSENGER-RNA
HISTONE DEMETHYLASES
MAXIMUM-LIKELIHOOD
Protein-Protein Interface Analysis and Hot Spots Identification for Chemical Ligand Design
期刊论文
current pharmaceutical design, 2014
Chen, Jing
;
Ma, Xiaomin
;
Yuan, Yaxia
;
Pei, Jianfeng
;
Lai, Luhua
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2015/11/13
Protein-protein interface analysis
small molecular binder
binding site detection
ligandability
hot spots
Pocket V.3
SMALL-MOLECULE INHIBITORS
DRUG DISCOVERY
BINDING-SITES
CONFORMATIONAL DYNAMICS
STRUCTURAL BIOLOGY
TRANSIENT POCKETS
PREDICTION
ALLOSTERY
DRUGGABILITY
MODULATION
De Novo Design of Multitarget Ligands with an Iterative Fragment-Growing Strategy
期刊论文
journal of chemical information and modeling, 2014
Shang, Erchang
;
Yuan, Yaxia
;
Chen, Xinyi
;
Liu, Ying
;
Pei, Jianfeng
;
Lai, Luhua
收藏
  |  
浏览/下载:2/0
  |  
提交时间:2015/11/10
HUMAN WHOLE-BLOOD
DRUG DISCOVERY
MULTIPLE LIGANDS
LEAD DISCOVERY
CYCLOOXYGENASE
INHIBITORS
BIOSYNTHESIS
NETWORK
BIOLOGY
Molecular docking and molecular dynamics studies on the structure-activity relationship of fluoroquinolone for the HERG channel
期刊论文
分子生物系统, 2014
Luo, Fang
;
Gu, Jiangyong
;
Chen, Lirong
;
Xu, Xiaojie
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2015/11/10
POLYMORPHIC VENTRICULAR-TACHYCARDIA
INTERVAL PROLONGATION
POTASSIUM CHANNEL
FREE-ENERGY
K+ CHANNEL
CARDIAC-ARRHYTHMIA
LIGAND-BINDING
QT INTERVAL
FORCE-FIELD
DRUG
Allosteric sites can be identified based on the residue-residue interaction energy difference
期刊论文
proteins, 2014
Ma Xiaomin
;
Qi Yifei
;
Lai Luhua
收藏
  |  
浏览/下载:4/0
  |  
提交时间:2015/11/11
CAVITY,MM/GBSA,allosteric site identification,energy decomposition,residue-residue interaction energy
Point Decoration of Silicon Nanowires: An Approach Toward Single- Molecule Electrical Detection**
期刊论文
angewandte chemie international edition, 2014
Wang, Jindong
;
Shen, Fangxia
;
Wang, Zhenxing
;
He, Gen
;
Qin, Jinwen
;
Cheng, Nongyi
;
Yao, Maosheng
;
Li, Lidong
;
Guo, Xuefeng
收藏
  |  
浏览/下载:7/0
  |  
提交时间:2015/11/11
biosensors
H1N1 antibody
point decoration
silicon nanowires
single-molecule studies
FIELD-EFFECT TRANSISTORS
WALLED CARBON NANOTUBES
HYDROGEN-TERMINATED SILICON
PROSTATE-SPECIFIC ANTIGEN
LABEL-FREE
REAL-TIME
ORGANIC MONOLAYERS
ELECTRONIC DEVICES
POROUS SILICON
BIOSENSORS
Ligand Clouds around Protein Clouds: A Scenario of Ligand Binding with Intrinsically Disordered Proteins
期刊论文
plos computational biology, 2013
Jin, Fan
;
Yu, Chen
;
Lai, Luhua
;
Liu, Zhirong
收藏
  |  
浏览/下载:3/0
  |  
提交时间:2015/11/10
SECONDARY STRUCTURE
ENERGY LANDSCAPE
CHEMICAL-SHIFTS
MYC-MAX
MOLECULAR SIMULATIONS
UNSTRUCTURED PROTEINS
TRANSCRIPTION FACTORS
COUPLED BINDING
PHYSICAL BASIS
C-MYC
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