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Role and Mechanism of the Interaction of BCR-ABL with E3 Ligase c-CBL in Targeting Therapy of Chronic Myelogenous Leukemia 期刊论文
Zhongguo shi yan xue ye xue za zhi, 2017, 卷号: 25, 期号: 1, 页码: 42-49
作者:  Mao, Jian-Hua;  Huang, Qiu-Hua;  Liu, Ping;  Luo, Cheng;  Xi, Xiao-Dong
收藏  |  浏览/下载:22/0  |  提交时间:2019/01/08
Discovery of novel Ponatinib analogues for reducing KDR activity as potent FGFRs inhibitors 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 126, 页码: 122-132
作者:  Liu, Yang;  Peng, Xia;  Guan, Xiaocong;  Lu, Dong;  Xi, Yong
收藏  |  浏览/下载:42/0  |  提交时间:2019/01/08
Role and Mechanism of the Interaction of BCR-ABL with E3 Ligase c-CBL in Targeting Therapy of Chronic Myelogenous Leukemia 期刊论文
Journal of Experimental Hematology, 2017, 卷号: 25, 期号: 1, 页码: 42-49
作者:  Mao Jianhua;  Huang Qiuhua;  Liu Ping;  Luo Cheng;  Xi Xiaodong
收藏  |  浏览/下载:32/0  |  提交时间:2019/01/08
BCR-ABL与泛素E3连接酶c-CBL的相互作用在慢性髓系白血病靶向治疗中的作用及相关机制研究 期刊论文
中国实验血液学杂志, 2017, 卷号: 025, 期号: 001, 页码: 42
作者:  毛建华;  黄秋花;  刘萍;  罗成;  奚晓东
收藏  |  浏览/下载:5/0  |  提交时间:2020/07/01
Identification of Bisindolylmaleimide IX as a potential agent to treat drug-resistant BCR-ABL positive leukemia 期刊论文
ONCOTARGET, 2016, 卷号: 7, 期号: 43, 页码: 69945-69960
作者:  Zhang, Xin;  Jia, Deyong;  Ao, Junping;  Liu, Huijuan;  Zang, Yi
收藏  |  浏览/下载:28/0  |  提交时间:2019/01/08
Y-632 inhibits heat shock protein 90 (Hsp90) function by disrupting the interaction between Hsp90 and Hsp70/Hsp90 organizing protein, and exerts antitumor activity in vitro and in vivo 期刊论文
CANCER SCIENCE, 2016, 卷号: 107, 期号: 6, 页码: 782-790
作者:  Wang, Wenqian;  Liu, Yang;  Zhao, Zhixin;  Xie, Chengying;  Xu, Yongping
收藏  |  浏览/下载:14/0  |  提交时间:2019/01/08
Dual Inhibition of Bcr-Abl and Hsp90 by C086 Potently Inhibits the Proliferation of Imatinib-Resistant CML Cells 期刊论文
CLINICAL CANCER RESEARCH, 2015, 卷号: 21, 期号: 4, 页码: 833-843
作者:  Wu, Lixian;  Yu, Jing;  Chen, Ruijia;  Liu, Yang;  Lou, Liguang
收藏  |  浏览/下载:37/0  |  提交时间:2019/01/08
Curcumin derivative C817 inhibits proliferation of imatinib-resistant chronic myeloid leukemia cells with wild-type or mutant Bcr-Abl in vitro 期刊论文
ACTA PHARMACOLOGICA SINICA, 2014, 卷号: 35, 期号: 3, 页码: 401-409
作者:  Wu, Li-xian;  Wu, Ying;  Chen, Rui-jia;  Liu, Yang;  Huang, Li-sen
收藏  |  浏览/下载:20/0  |  提交时间:2019/01/08
Flumatinib, a selective inhibitor of BCR-ABL/PDGFR/KIT, effectively overcomes drug resistance of certain KIT mutants 期刊论文
CANCER SCIENCE, 2014, 卷号: 105, 期号: 1, 页码: 117-125
作者:  Zhao, Jie;  Quan, Haitian;  Xu, Yongping;  Kong, Xiangqian;  Jin, Lu
收藏  |  浏览/下载:27/0  |  提交时间:2019/01/08
Design, Synthesis, and Biological Evaluation of Novel Conformationally Constrained Inhibitors Targeting Epidermal Growth Factor Receptor Threonine(790) -> Methionine(790) Mutant 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2012, 卷号: 55, 期号: 6, 页码: 2711-2723
作者:  Chang, Shaohua;  Zhang, Lianwen;  Xu, Shilin;  Luo, Jinfeng;  Lu, Xiaoyun
收藏  |  浏览/下载:18/0  |  提交时间:2019/01/08


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