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A Peptide Binder of E3 Ligase Adaptor SPOP Disrupts Oncogenic SPOP-Protein Interactions in Kidney Cancer Cells 期刊论文
CHINESE JOURNAL OF CHEMISTRY, 2020, 页码: 274-280
作者:  Wang, Zhen;  Zhang, Hao;  Chen, Baoen;  Ouyang, Sisheng;  Zheng, Tong
收藏  |  浏览/下载:124/0  |  提交时间:2021/05/24
Targeted Proteomics Combined with Affinity Mass Spectrometry Analysis Reveals Antagonist E7 Acts As an Intracellular Covalent Ligand of Orphan Receptor GPR52 期刊论文
ACS CHEMICAL BIOLOGY, 2020, 卷号: 15, 期号: 12, 页码: 3275-3284
作者:  Ma, Mengna;  Guo, Shimeng;  Lin, Xi;  Li, Shanshan;  Wu, Yiran
收藏  |  浏览/下载:16/0  |  提交时间:2021/05/24
Small molecules targeting the innate immune cGAS-STING-TBK1 signaling pathway 期刊论文
ACTA PHARMACEUTICA SINICA B, 2020, 卷号: 10, 期号: 12, 页码: 2272-2298
作者:  Ding, Chunyong;  Song, Zilan;  Shen, Ancheng;  Chen, Tingting;  Zhang, Ao
收藏  |  浏览/下载:23/0  |  提交时间:2021/05/24
The Active Constituent From Gynostemma Pentaphyllum Prevents Liver Fibrosis Through Regulation of the TGF-beta 1/NDRG2/MAPK Axis 期刊论文
FRONTIERS IN GENETICS, 2020, 卷号: 11, 页码: 11
作者:  Huang, Hui;  Wang, Kuifeng;  Liu, Qian;  Ji, Feihong;  Zhou, Hu
收藏  |  浏览/下载:32/0  |  提交时间:2020/12/24
The novel small-molecule TPN10456 inhibits Th17 cell differentiation and protects against experimental autoimmune encephalomyelitis 期刊论文
CELLULAR & MOLECULAR IMMUNOLOGY, 2020, 页码: 4
作者:  Yang, Cuixia;  Lv, Jie;  Jiang, Xiangrui;  Xiang, Zhenglong;  Gong, Ran
收藏  |  浏览/下载:22/0  |  提交时间:2020/12/24
Engineering Prodrug Nanomedicine for Cancer Immunotherapy 期刊论文
ADVANCED SCIENCE, 2020, 页码: 33
作者:  Yang, Bin;  Gao, Jing;  Pei, Qing;  Xu, Huixiong;  Yu, Haijun
收藏  |  浏览/下载:20/0  |  提交时间:2020/12/21
SOMCL-863, a novel, selective and orally bioavailable small-molecule c-Met inhibitor, exhibits antitumor activity both in vitro and in vivo (vol 351, pg 413, 2014) 期刊论文
CANCER LETTERS, 2020, 卷号: 486, 页码: 71-72
作者:  Wang, Lu;  Ai, Jing;  Shen, Yanyan;  Zhang, Haotian;  Peng, Xia
收藏  |  浏览/下载:10/0  |  提交时间:2020/12/24
Tideglusib and Its Analogues As Inhibitors of Staphylococcus aureus SrtA 期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2020, 卷号: 63, 期号: 15, 页码: 8442-8457
作者:  Yang, Teng;  Zhang, Tao;  Guan, Xiang-Na;  Dong, Ze;  Lan, Lefu
收藏  |  浏览/下载:20/0  |  提交时间:2020/12/24
Structural insights into the activation of GLP-1R by a small molecule agonist 期刊论文
CELL RESEARCH, 2020, 页码: 3
作者:  Ma, Honglei;  Huang, Wei;  Wang, Xiaoxi;  Zhao, Lihua;  Jiang, Yi
收藏  |  浏览/下载:38/0  |  提交时间:2020/12/24
Targeting FTO Suppresses Cancer Stem Cell Maintenance and Immune Evasion 期刊论文
CANCER CELL, 2020, 卷号: 38, 期号: 1, 页码: 79-+
作者:  Su, Rui;  Dong, Lei;  Li, Yangchan;  Gao, Min;  Han, Li
收藏  |  浏览/下载:33/0  |  提交时间:2020/12/24


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