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科研机构
合肥物质科学研究院 [10]
上海药物研究所 [9]
高能物理研究所 [3]
厦门大学 [2]
北京大学 [2]
兰州理工大学 [2]
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期刊论文 [32]
学位论文 [2]
发表日期
2017 [34]
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PI-273, a Substrate-Competitive, Specific Small-Molecule Inhibitor of PI4KII alpha, Inhibits the Growth of Breast Cancer Cells
期刊论文
CANCER RESEARCH, 2017, 卷号: 77, 期号: 22, 页码: 6253-6266
作者:
Li, Jiangmei
;
Gao, Zhen
;
Zhao, Dan
;
Zhang, Lunfeng
;
Qiao, Xinhua
收藏
  |  
浏览/下载:24/0
  |  
提交时间:2019/01/08
Structure-based design and synthesis of 2,4-diaminopyrimidines as EGFR L858R/T790M selective inhibitors for NSCLC
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 140, 页码: 510-527
作者:
Chen, Lingfeng
;
Fu, Weitao
;
Feng, Chen
;
Qu, Rong
;
Tong, Linjiang
收藏
  |  
浏览/下载:55/0
  |  
提交时间:2019/01/08
Epidermal growth factor receptor
Tyrosine kinase inhibitors
Non-small cell lung cancer
T790M
Mutant-selective
Discovery, mechanism and metabolism studies of 2,3-difluorophenyl-linker-containing PARP1 inhibitors with enhanced in vivo efficacy for cancer therapy
期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 138, 页码: 514-531
作者:
Chen, Wenhua
;
Guo, Ne
;
Qi, Minghui
;
Dai, Haiying
;
Hong, Minghuang
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  |  
浏览/下载:30/0
  |  
提交时间:2019/01/08
Antitumor drug
BRCA1/2
PARP inhibitors
Molecular docking
Targeted delivery of sirna using rgdfc-conjugated functionalized selenium nanoparticles for anticancer therapy
期刊论文
Journal of materials chemistry b, 2017, 卷号: 5, 期号: 33, 页码: 6941-6952
作者:
Xia, Yu
;
Lin, Zhengfang
;
Li, Yinghua
;
Zhao, Mingqi
;
Wang, Changbing
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  |  
浏览/下载:32/0
  |  
提交时间:2019/05/08
Cyanobacterial peptides as a prototype for the design of cathepsin D inhibitors
期刊论文
JOURNAL OF PEPTIDE SCIENCE, 2017, 卷号: 23, 期号: 9, 页码: 701-706
作者:
Xu, Hao
;
Bao, Keting
;
Tang, Shuai
;
Ai, Jing
;
Hu, Haiyan
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  |  
浏览/下载:26/0
  |  
提交时间:2019/01/08
cathepsin D
inhibitor
peptides
structural modification
transition-state mimics
Pathological expression of tissue factor confers promising antitumor response to a novel therapeutic antibody SC1 in triple negative breast cancer and pancreatic adenocarcinoma
期刊论文
ONCOTARGET, 2017, 卷号: 8, 期号: 35, 页码: 59086-59102
作者:
Zhang, Xuesai
;
Li, Qingrou
;
Zhao, Hui
;
Ma, Lanping
;
Meng, Tao
收藏
  |  
浏览/下载:33/0
  |  
提交时间:2019/01/08
tissue factor
triple negative breast cancer
pancreatic adenocarcinoma
metastasis
antibody-drug conjugate
Design, Synthesis and Anti-Proliferative Activities of 2,6-Substituted Thieno[3,2-d] pyrimidine Derivatives Containing ElectrophilicWarheads
期刊论文
MOLECULES, 2017, 卷号: 22, 期号: 5
作者:
Zhang, Qiumeng
;
Hu, Zonglong
;
Shen, Qianqian
;
Chen, Yi
;
Lu, Wei
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  |  
浏览/下载:15/0
  |  
提交时间:2019/01/08
thieno[3,2-d] pyrimidines
antitumor activities
acrylamide warheads
Synthesis and cytotoxic activity of novel tetrahydrobenzodifuran-imidazolium salt derivatives
期刊论文
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017, 卷号: 27, 期号: 8, 页码: 1808-1814
作者:
Zhang, Chao-Bo
;
Liu, Yang
;
Liu, Zheng-Fen
;
Duan, Sheng-Zu
;
Li, Min-Yan
收藏
  |  
浏览/下载:25/0
  |  
提交时间:2017/06/30
Tetrahydrobenzodifurans
Imidazolium salts
Cytotoxic activity
Cell cycle
Apoptosis
Discovery of (R)-1-(3-(4-Amino-3-(3-chloro-4-(pyridin-2-ylmethoxy)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one (CHMFL-EGFR-202) as a Novel Irreversible EGFR Mutant Kinase Inhibitor with a Distinct Binding Mode
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 7, 页码: 2944-2962
作者:
Wang, Aoli
;
Li, Xixiang
;
Wu, Hong
;
Zou, Fengming
;
Yan, Xiao-E
收藏
  |  
浏览/下载:34/0
  |  
提交时间:2018/07/26
Discovery of (R)-1-(3-(4-Amino-3-(3-chloro-4-(pyridin-2-ylmethoxy)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one (CHMFL-EGFR-202) as a Novel Irreversible EGFR Mutant Kinase Inhibitor with a Distinct Binding Mode
期刊论文
JOURNAL OF MEDICINAL CHEMISTRY, 2017, 卷号: 60, 期号: 7, 页码: 2944-2962
作者:
Wang, Aoli
;
Li, Xixiang
;
Wu, Hong
;
Zou, Fengming
;
Yan, Xiao-E
收藏
  |  
浏览/下载:41/0
  |  
提交时间:2018/07/26
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