Synthesis and Insecticidal Activity of N-tert-Butyl-N,N '-diacylhydrazines Containing 1,2,3-Thiadiazoles

doi:10.1021/jf104004q

	Synthesis and Insecticidal Activity of N-tert-Butyl-N,N '-diacylhydrazines Containing 1,2,3-Thiadiazoles
	Wang, Huan 1; Yang, Zhikun 1; Fan, Zhijin 1; Wu, Qingjun 2; Zhang, Youjun 2; Mi, Na 1; Wang, Shouxin 1; Zhang, Zhengcai 1; Song, Haibin 1; Liu, Feng 2
刊名	JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY
	2011
卷号	59 期号:2 页码:628-634
关键词	4-Methyl-1,2,3-thiadiazole diacylhydrazine Insect growth regulator
ISSN号	0021-8561
DOI	10.1021/jf104004q
通讯作者	Wang, Huan
英文摘要	N-tert-Butyl-N,N'-diacylhydrazines are nonsteroidal ecdysone agonists used as environmental benign pest regulators. In this paper, two series of new N-tert-butyl-N,N'-diacylhydrazine derivatives containing 1,2,3-thiadiazole were designed and synthesized. All structures of the synthesized compounds were confirmed by proton nuclear magnetic resonance ((1)H NMR), infrared spectroscopy (IR), and high-resolution mass spectrometry (HRMS). Bioasssay results indicated that most of the synthesized compounds possessed good insecticidal activities against Plutella xylostella L. and Culex pipiens pallens as compared with the positive control, tebufenozide. The results of this study indicated that 1,2,3-thiadiazoles, as an important active substructure, could improve or maintain the activity of the dicylhydrazines and favor novel pesticide development.
学科主题	Agriculture, Multidisciplinary ; Chemistry, Applied ; Food Science & Technology ; AGRICULTURE, MULTIDISCIPLINARY ; CHEMISTRY, APPLIED ; FOOD SCIENCE & TECHNOLOGY
语种	英语
出版者	AMER CHEMICAL SOC
WOS记录号	WOS:000286176100023
内容类型	期刊论文
源URL	[http://111.203.20.206/handle/2HMLN22E/101162]
专题	蔬菜花卉研究所_植物保护研究室
作者单位	1.Nankai Univ, State Key Lab Elementoorgan Chem, Tianjin 300071, Peoples R China 2.Chinese Acad Agr Sci, Inst Vegetables & Flowers, Beijing 100081, Peoples R China
推荐引用方式 GB/T 7714	Wang, Huan,Yang, Zhikun,Fan, Zhijin,et al. Synthesis and Insecticidal Activity of N-tert-Butyl-N,N '-diacylhydrazines Containing 1,2,3-Thiadiazoles[J]. JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY,2011,59(2):628-634.
APA	Wang, Huan.,Yang, Zhikun.,Fan, Zhijin.,Wu, Qingjun.,Zhang, Youjun.,...&Liu, Feng.(2011).Synthesis and Insecticidal Activity of N-tert-Butyl-N,N '-diacylhydrazines Containing 1,2,3-Thiadiazoles.JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY,59(2),628-634.
MLA	Wang, Huan,et al."Synthesis and Insecticidal Activity of N-tert-Butyl-N,N '-diacylhydrazines Containing 1,2,3-Thiadiazoles".JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY 59.2(2011):628-634.